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4-chloro-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[(4-methoxyphenyl)methyl]-N-(3-methoxypropyl)-1-methylazepane-2-carboxamide
3-(2-methoxyphenyl)-5-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2,4-oxadiazole
N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
N-(2,5-difluorophenyl)-3-(isoquinolin-5-ylformamido)propanamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[(2,2-dimethyloxan-4-yl)methyl]piperidin-4-yl}propanamide
1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
3-(5-{2-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
2-(3-fluorophenyl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]azepane
N-ethyl-4-hydroxy-1-methyl-N-[2-(4-methylbenzenesulfonyl)ethyl]piperidine-4-carboxamide
2-({[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl]amino}methyl)-4-methoxyphenol
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-3-acetamidopyrrolidine-1-carboxamide
[1-(3-methoxyphenyl)ethyl](methyl){[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1S,4S)-2-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}-2,5-diazabicyclo[2.2.1]heptane
5-fluoro-N,1,3-trimethyl-N-(3-phenoxypropyl)-1H-indole-2-carboxamide
N-(3-{[(4-fluorophenyl)methyl]sulfanyl}propyl)oxolane-3-carboxamide
N-(cyclopropylmethyl)-N-(2-methoxyethyl)-4-methylpyrimidine-5-carboxamide
2,4-dimethoxy-6-(1H-pyrazol-3-yl)-1,3,5-triazine
[1-(6-ethyl-2-methylquinoline-4-carbonyl)azepan-2-yl]methanol
4-[3-(furan-2-yl)phenyl]-1-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole
2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-[2-(pyrazin-2-yl)ethyl]acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N,2-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-[(3-chlorophenyl)methyl]-N-propyl-2-(pyridin-2-yl)acetamide
2-amino-4-[2-(dimethylamino)-1,3-thiazol-5-yl]-6-methyl-5,6,7,8-tetrahydroquinoline-3-carbonitrile
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(4-hydroxyphenyl)methyl]pyrrolidine-2-carboxylate
3-hydroxy-1-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-2-(1,3-thiazol-2-yl)piperidine
5-(4-benzylpiperidin-1-yl)-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole
(1s,4s)-4-hydroxy-N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]cyclohexane-1-carboxamide
N-({5-[4-(dimethylamino)pyrimidin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(5-ethylthiophene-2-carbonyl)pyrrolidin-3-yl]methanol
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
propyl N-{[(3S,4S)-1-(3-aminobenzoyl)-3-hydroxypiperidin-4-yl]methyl}carbamate
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
3-{1-[(5-cyclopentylthiophen-2-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
2-chloro-6-fluoro-3-methyl-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]benzamide
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
2-{3-[(3-chlorophenyl)methyl]-5-(2,6-dimethylpyrimidin-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidin-3-ol
1-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
4-benzyl-3-ethyl-1-(5-methoxy-4-oxo-1,4-dihydropyridine-2-carbonyl)-1,4-diazepan-5-one
(1S,3R)-3-amino-N-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]phenyl}cyclopentane-1-carboxamide
{2-[4-(5-ethyl-2-methylpyrimidin-4-yl)morpholin-2-yl]ethyl}dimethylamine
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-methoxybutan-1-one
1-ethyl-3,5-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1H-pyrazole-4-carboxamide
5-{4-[3-(1,3-benzothiazol-2-yl)propanoyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
1-[1-(4-fluorophenyl)-2,2-dimethylcyclopropaneamido]cycloheptane-1-carboxamide
N-(2-methoxyethyl)-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide