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3-[4-(2-methylphenyl)-1H-pyrazol-5-yl]-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidine
3-amino-3-(3,4-dimethoxyphenyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
[(3R,4R)-1-(2-chloro-5-fluorobenzoyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
1-(5-chloro-2-methylphenyl)-4-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
1-{1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]azetidin-3-yl}-2-methylpiperidine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(3-phenyl-1,2-oxazole-5-carbonyl)pyrrolidin-3-yl]methanol
5-methyl-3-{5-[5-(oxolan-2-yl)thiophene-2-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-1,2-oxazole
N-(3,4-dimethoxyphenyl)-1-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]piperidin-3-amine
8-(dimethyl-1,3-thiazole-5-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-[3-(methoxymethyl)pyrrolidin-1-yl]-5-(naphthalen-1-yl)-1,2,4-triazine
N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-N-methyl-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
6-oxo-1-(3-phenylpropyl)-N-[3-(pyridin-3-yloxy)propyl]piperidine-3-carboxamide
N-cyclopropyl-4-(1H-pyrazol-1-yl)-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}benzamide
4-{1-[1-(6-methylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
(1R,3S)-7-(2,1,3-benzoxadiazol-4-ylmethyl)-3-[2-(dimethylamino)ethoxy]-7-azaspiro[3.5]nonan-1-ol
9-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-2,3,4,9-tetrahydro-1H-carbazole-7-carboxamide
6,8-dimethyl-3-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-ethyl-N-methylacetamide
1-[2-(benzyloxy)phenyl]-3-methyl-3-(1-methylpyrrolidin-3-yl)urea
1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pent-4-en-1-one
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]propan-1-one
ethyl 1-[3-(1,2-oxazinan-2-yl)propanoyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-(4-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrazine
1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-N-[2-(pyrrolidin-1-yl)ethyl]piperidine-3-carboxamide
1-(2-methoxybenzoyl)-4-(3-propyl-1H-pyrazole-5-carbonyl)piperazine
2-{[(4-chlorophenyl)methyl]amino}-N-[(2-fluorophenyl)methyl]acetamide
4-methoxy-2-[(3-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidin-1-yl)methyl]phenol
N-methyl-3-{[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
2-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-benzyl-8-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
N-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-N-(3-methylphenyl)methanesulfonamide
3-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-4-methylpyridine
2-({[(3R,4R)-4-(hydroxymethyl)-1-[(6-methylquinolin-5-yl)methyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
ethyl 4-[(1-{4-[2-(3-fluorophenyl)acetamido]phenyl}piperidin-4-yl)amino]piperidine-1-carboxylate
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H-indazole-3-carboxamide
3-(2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
(4aS,7aR)-1-[(2-ethoxyphenyl)methyl]-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(6-cyanopyridin-3-yl)-3-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)urea
(3S,4S)-1-[6-(methoxymethyl)pyrimidin-4-yl]-4-propylpyrrolidine-3-carboxylic acid
4-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-3-butyl-1-methylpiperazin-2-one
4-{1-[(4-phenylphenyl)methyl]-1H-1,2,3,4-tetrazol-5-yl}-1,4-oxazepan-6-ol
3-chloro-N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]pyridine-4-carboxamide
N-(1-{7-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
1-[1-(2,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
2-(2,4-dichlorophenoxy)-N-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide