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N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-methyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}thieno[2,3-d]pyrimidin-4-amine
5-[5-(2-ethoxyethyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-(morpholin-4-yl)benzamide
2-(2-methoxyethyl)-9-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-4-methylpentan-1-one
{1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}(pyridin-2-yl)methanol
4-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methyl-1H-1,3-benzodiazole
2-[2-(1H-imidazol-1-yl)ethyl]-1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(methylsulfanyl)acetamide
(3aS,6aS)-2-cyclohexyl-5-[(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-methyl-6-(propan-2-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-6-methyl-4-oxo-4H-pyran-2-carboxamide
3-acetyl-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]benzamide
N-(3-chloro-2-methylphenyl)-3-(4-phenylpiperazin-1-yl)piperidine-1-carboxamide
3-(oxolan-3-yl)-5-[4-(1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazole
3-[(3R,4S)-1-[4-(dimethylamino)benzoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(5S,9aS,9bS)-2-(2-methoxyphenyl)-5-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[2-(pyridin-3-yl)piperidine-1-carbonyl]-6-(4H-1,2,4-triazol-4-yl)pyridine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethan-1-one
6-(8-methoxy-2-methylquinolin-5-yl)-2-methyl-2,3-dihydropyridazin-3-one
1-methyl-3-[5-(2-methylbutan-2-yl)-1,3,4-thiadiazol-2-yl]-1-(thiophen-2-ylmethyl)urea
N-(1-cycloheptylpiperidin-3-yl)pyridine-4-carboxamide
(1S,5R)-6-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
2-{1-[(2,6-difluoro-3-methoxyphenyl)methyl]azetidin-3-yl}-1H-1,3-benzodiazole
N-[(3R,5S)-1-(3-hydroxypropyl)-5-(methylcarbamoyl)pyrrolidin-3-yl]-5-methoxy-1H-indole-2-carboxamide
2-(3-hydroxypropyl)-9-(5-methylpyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(thiophen-2-yl)propan-2-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
N-{4-[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]phenyl}-3,4-dimethylpiperazine-1-carboxamide
4-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-(methylsulfanyl)-1,3-thiazole
(4aS,8aR)-6-(1H-indol-2-ylmethyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
N-(1,4-dioxan-2-ylmethyl)-N-methyl-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-[(2-methylphenyl)methyl]-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3R,4S)-1-(2,3-dichlorobenzoyl)-3,4-dimethylpiperidin-4-ol
1-cyclopentyl-4-[2-(methylsulfanyl)benzoyl]-1,4-diazepane
1-(3-hydroxyphenyl)-4-[1-(2-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
2-[(2R)-3-hydroxy-2-methylpropyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(1-{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)methanesulfonamide
2,2-diphenyl-1-{4-[1-(propan-2-yl)piperidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}ethan-1-ol
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(pyrimidin-2-yl)piperidin-3-yl]propan-1-ol
1-ethyl-4-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
4-{5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}morpholine
(3aS,6aS)-2-(ethanesulfonyl)-5-[4-(methylamino)pyrimidin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-[4-amino-6-(benzylamino)-1,3,5-triazin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
6-fluoro-2-({4-[(1-methylpiperidin-3-yl)methyl]piperazin-1-yl}methyl)quinolin-4-ol
4,6-dimethyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-ethyl-N-(oxan-4-ylmethyl)-3-(piperidin-4-ylmethyl)benzamide
1-(4-methoxyphenyl)-3-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-3-methylurea
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carbonitrile
3-(azepane-1-sulfonyl)-5-(3-methyl-1H-pyrazol-1-yl)benzoic acid