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(2S)-2-{[(2-chloro-5-fluorophenyl)carbamoyl]amino}-3-methylbutanamide
N-cyclopropyl-5-(1-methylpiperidine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
N2,N2-dimethyl-N4-[3-methyl-1-(pyridin-3-yl)butyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-[1-(2-phenylethyl)-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperazin-2-yl]ethan-1-ol
(3S,4R)-1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N-{[2-(4-chlorophenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)acetamide
(3aS,6aS)-5-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-N,N-dimethylpyridine-3-carboxamide
1-(4-{[(cyclobutylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-2-(1H-indazol-3-yl)-N-methylacetamide
methyl 4-(methylsulfanyl)-2-{[2-(3-phenylpropyl)-1,3-benzoxazol-5-yl]formamido}butanoate
N-{1-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylpyridine-2-carboxamide
1-cyclopentyl-4-(6-oxo-1,6-dihydropyridine-2-carbonyl)piperazin-2-one
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
8-{thieno[2,3-d]pyrimidin-4-yl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
methyl (1R,3S,3aR,6aS)-5-benzyl-3-(2-methylphenyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1,7-dimethyl-2-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1H-indole
5-[3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]pyrazin-2-ol
2-methyl-5-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}pyrimidin-4-ol
2-methyl-6-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]phenol
(2S)-1-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}-4-methyl-2-phenylpiperazine
1-(2-{9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-oxoethyl)-4-phenylpyrrolidin-2-one
N-ethyl-6-(3-fluorophenyl)-N-[(1-methylpyrrolidin-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[2-hydroxy-2-(pyridin-2-yl)ethyl]-3,4,7-trimethyl-1H-indole-2-carboxamide
1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
4-[4-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-2-methyl-1,2-dihydrophthalazin-1-one
6-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-methyl-N-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
3-[(dimethylamino)methyl]-1-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}pyrrolidin-3-ol
1-(furan-2-yl)-2-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethane-1,2-dione
1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(thian-4-yl)piperazine
1-[2-(propan-2-yloxy)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(3aR,7aS)-2-(5-propyl-1,3,4-oxadiazole-2-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-(2-chloro-4-fluorophenyl)-1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]ethan-1-one
N-[3-(4-cyclopentyl-1,4-diazepan-1-yl)-3-oxopropyl]-N-methylmethanesulfonamide
(3S,4S)-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrrolidin-3-ol
4-{[3,3-dimethyl-1-(pyrrolidin-1-yl)butan-2-yl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
5-(4-acetylphenoxymethyl)-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
2-methyl-5-(2-{2-[(9H-purin-6-yl)amino]ethyl}morpholin-4-yl)-2,3-dihydropyridazin-3-one
(3R,4S)-4-cyclopropyl-1-[3-(2-ethoxyethoxy)benzoyl]pyrrolidin-3-amine
N,N-dimethyl-2-phenyl-2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)acetamide
N-{4-[3-methyl-4-(propan-2-yl)piperazine-1-carbonyl]phenyl}ethane-1-sulfonamide
3-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]-2,8-diazaspiro[4.5]decane
(4aR,7aS)-1-acetyl-4-[(1-methyl-1H-imidazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopentyl-4-[4-({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)piperidin-1-yl]benzamide
2-(ethylamino)-N-[3-(morpholin-4-yl)propyl]pyrimidine-5-carboxamide
6-(4-chlorophenyl)-N-(1,4-dioxan-2-ylmethyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
methyl 3-(furan-2-amido)-5-[(3-hydroxy-3-methylbutan-2-yl)amino]-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-methyl-1-(2-phenylethyl)-5-[(propan-2-yl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide