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N-(cyclohex-1-en-1-ylmethyl)-8-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(3R,4R)-4-(azepan-1-yl)-1-[1-(3-methoxyphenyl)piperidin-4-yl]piperidin-3-ol
4-[({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)methyl]-1-(2-methoxyethyl)pyrrolidin-2-one
1-(2,1,3-benzothiadiazol-5-ylmethyl)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidine-3-carboxamide
2-(morpholin-4-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]-2-(pyridin-3-yl)ethan-1-one
(1S,6R)-9-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[(5-methylpyrazin-2-yl)methyl]-8-(oxane-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(2R,3R)-3-{methyl[2-(4-methylphenoxy)ethyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[2-(2-fluorophenyl)ethyl]-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidine
1-ethyl-4-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N-(butan-2-yl)-5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole
1-(1,3-dioxo-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindol-4-yl)-N-(propan-2-yl)piperidine-3-carboxamide
(1S,5R)-6-(1-ethyl-1H-pyrazole-4-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
5-{[methyl({[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}-N-propylpyrimidin-2-amine
2-(1-methylpyrrolidin-3-yl)-9-(1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-{1-[2-(4-fluorophenyl)-2-hydroxyacetyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
1-(1'-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
(1R,5R)-6-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
methyl (2R)-2-({2-[(quinolin-6-yloxy)methyl]-1,3-oxazol-4-yl}formamido)propanoate
2-(ethylamino)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]pyrimidine-5-carboxamide
3-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
1-{2-methylthieno[2,3-d]pyrimidin-4-yl}-4-(oxan-4-yl)piperazine
N-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-2-phenylethyl}-N,2-dimethylfuran-3-carboxamide
1-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]azepane
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
N,N-dimethyl-1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}pyrrolidin-3-amine
N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-4-ylmethyl)cycloheptanecarboxamide
2-amino-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}-4-phenylpyrimidine-5-carboxamide
2-cyano-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)benzamide
7-(2,1,3-benzoxadiazol-4-ylmethyl)-2-oxa-7-azaspiro[4.5]decane
[2-(2-aminopyrimidin-5-yl)phenyl]methanol
6-{methyl[2-(methylsulfanyl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-(3-hydroxy-4-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1-ethyl-1H-indazol-3-yl)methyl]-2-(1-ethylpiperidin-4-yl)acetamide
2-methoxy-4-[4-(2-methoxyethoxy)phenyl]pyridine-3-carbonitrile
5-ethyl-N4-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrimidine-2,4-diamine
2-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-N-[(5-methylfuran-2-yl)methyl]quinazolin-4-amine
1-[2-(2-methoxy-2-methylpropyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-(2-phenylethyl)piperidine-3-carboxamide
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
2-(3,4-dichlorophenyl)-4-(5,6-dimethylpyrimidin-4-yl)morpholine
(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
N-ethyl-4-fluoro-N-(1-hydroxypropan-2-yl)-3-methylbenzamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(2-phenylacetyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
4-(4-{[(5-methylpyrazin-2-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
(4S)-1-{3-[(dimethylamino)methyl]benzoyl}-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
4-(4-fluorophenyl)-1-[4-(pyridin-2-yl)pyrimidin-2-yl]piperidin-4-ol
[(3R,4S)-1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
6-{1-oxaspiro[4.4]nonan-3-yl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
[3-(4-phenyl-1H-imidazol-5-yl)phenyl]methanol