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N-{4-methyl-2-[3-(1H-pyrazol-3-yl)phenyl]phenyl}propanamide
1-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(2-hydroxy-3-methoxypropyl)-4-{[(4-methylphenyl)amino]methyl}benzamide
8-(6-aminopyrimidin-4-yl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{5-[5-(4-methoxyphenyl)furan-2-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
3-({[3-(4-methyl-1,3-thiazol-5-yl)propyl]amino}methyl)piperidin-3-ol
methyl 6-[(4-methoxy-2,3-dimethylphenyl)methyl]-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N4-ethyl-N2-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]pyrimidine-2,4-diamine
1-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]-4-(2-methylphenoxy)piperidine-4-carboxylic acid
1-(2-fluorophenyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]cyclopropane-1-carboxamide
N-{3-[(pyridin-3-yl)amino]propyl}-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
2,3-dimethyl-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]quinoxaline-6-carboxamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-(thiophen-2-yl)acetamide
5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-2,2-dimethylthiomorpholin-3-one
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-methoxypropan-1-one
(4aS,8aR)-6-(furan-2-ylmethyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}quinoline-4-carboxamide
N-(1-{7-[3-(2-chlorophenyl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)oxolane-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(1H-indol-2-ylformamido)acetic acid
[(2S,6S)-4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
(2S)-2-acetamido-N,4-dimethyl-N-(quinolin-5-ylmethyl)pentanamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(pyridin-3-yl)pyrimidine
N-[(3S,7S,8aS)-3-[(4-chlorophenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorobenzamide
methyl 1-[(3-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-4-methoxyphenyl)methyl]piperidine-4-carboxylate
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-methyl-9-(4-methylpyridine-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-4-(pyrrolidin-1-yl)butan-1-one
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
(3S,4R)-1-(3-chloro-5-methoxybenzoyl)-3-methoxypiperidin-4-amine
2-(2,2-diphenylacetyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
ethyl 1-(1,3-benzothiazol-2-yl)-5-({[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-1H-pyrazole-4-carboxylate
(1R,3S,5S)-8-(3-{[(4-methylphenyl)methyl]amino}benzoyl)-8-azabicyclo[3.2.1]octan-3-ol
4-methyl-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1,2,3-thiadiazole-5-carboxamide
2-phenyl-1-[1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-4-yl]ethan-1-ol
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
3-[(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)methyl]benzoic acid
(3S,4R)-1-(4-fluoro-3-methylbenzoyl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
4-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(4-methylpentyl)morpholine
5-fluoro-2-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
4-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
4-fluoro-N-[2-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]benzamide
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
4-benzyl-1-methyl-3-[1-(3-methylpyridine-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,4S)-2-(3-chloro-4-methoxyphenyl)-5-[1-(2-phenylethyl)piperidin-4-yl]-2,5-diazabicyclo[2.2.1]heptan-3-one
2-(1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-4-methyl-1H-1,3-benzodiazole
1-(4-ethoxy-3-methylphenyl)-4-[2-(pyridin-2-yl)pyrrolidin-1-yl]butane-1,4-dione
N-cyclohexyl-N,4-dimethyl-5-{1-[(thian-4-yl)amino]ethyl}pyrimidin-2-amine