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2-[5-(6-chloro-1,3-benzothiazol-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
1-(4-{[(1R)-1-cyclohexylethyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-[4-(adamantan-1-yl)piperazin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
5-ethyl-2-({4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridine
2-({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
6-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)pyridine-2-carboxylic acid
5-ethyl-2-[4-(pyridin-4-yl)piperazin-1-yl]pyrimidine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}propanamide
3-cyclohexyl-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-1H-pyrazole-4-carboxamide
9-(2-oxoimidazolidine-4-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(hydroxymethyl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
N,2-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[2-(4-fluorophenyl)piperidin-1-yl]propan-1-one
1-(4-benzylpiperazin-1-yl)-3-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-yl]propan-1-one
7-[2-(2,5-dimethoxyphenyl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-(cyclopropylmethyl)-8-(2-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
2-ethoxy-5-[2-(3-methylpiperazin-1-yl)pyrimidin-4-yl]benzoic acid
(4aS,8aR)-1-propyl-6-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}-decahydro-1,6-naphthyridin-2-one
(4S,4aS,8aS)-4-phenyl-1-(1H-pyrrole-3-carbonyl)-decahydroquinolin-4-ol
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-[4-(5-methyl-1,2-oxazole-3-carbonyl)morpholin-3-yl]acetamide
3-({2-[1-(thiophene-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
(3S,4S)-1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(propan-2-yloxy)pyrrolidin-3-ol
N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanamide
7-methanesulfonyl-N4-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-[2-(3-fluorophenyl)ethyl]-4-{4-[(3,4,5-trimethoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-methyl-9-(1,3-thiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[3-phenyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
N-[2-(4-fluorophenyl)-2-(piperidin-1-yl)ethyl]-4-hydroxy-1-methylpiperidine-4-carboxamide
N,N-dimethyl-5-(1-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-imidazol-2-yl)pyridin-2-amine
N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]acetamide
2-{4-[1-(3-methylpyridin-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}-1-(morpholin-4-yl)ethan-1-one
(1R,3S)-3-methoxy-7-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
3-{2-[benzyl(3-hydroxy-2-methylpropyl)amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
(1R,7S)-N-methyl-4-oxo-3-(2-phenoxyethyl)-N-(1H-pyrazol-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-ethyl-4-methyl-N-[(3R,4S)-1-(oxan-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-1,3-oxazole-5-carboxamide
N-{[4-(dimethylsulfamoyl)phenyl]methyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetic acid
9-{[4-(2-aminoethyl)phenyl]methyl}-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
(1R,6S)-9-methyl-3-(1H-pyrazole-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-[2-(4-methoxyphenyl)ethyl]piperidine-1-carboxamide
1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one
3-[4-(3-methoxyphenyl)-2-methyl-5-oxopiperazine-1-carbonyl]-1,2-dihydroquinoxalin-2-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
2-[(furan-2-ylmethyl)({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amino]butan-1-ol
3-phenyl-5-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-2-yl)-1,2,4-oxadiazole
(3S,4S)-1-[2-(methylamino)pyridine-3-carbonyl]-4-(naphthalen-2-yl)piperidin-3-ol
2,3-dimethoxy-N-[5-methyl-2-(2-methylbenzamido)phenyl]benzamide
6-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
8-chloro-2-(furan-2-yl)-N-(1,2-oxazol-3-ylmethyl)quinoline-4-carboxamide