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3-(1H-imidazol-1-ylmethyl)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine
(3S,4R)-1-({[(5-carboxyfuran-2-yl)methyl]carbamoyl}methyl)-4-phenylpyrrolidine-3-carboxylic acid
(3R)-1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}pyrrolidin-3-ol
7-({3-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxa-7-azaspiro[4.5]decan-8-one
5-(3,3-diphenylpiperidine-1-carbonyl)pyrazin-2-ol
2-[2-(1H-imidazol-4-yl)ethyl]-8-(2-phenylacetyl)-2,8-diazaspiro[5.5]undecan-3-one
3-methyl-1-(1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)butan-1-ol
1-[(3R,4R)-3-hydroxy-4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
4-(furan-3-ylmethyl)-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(azonan-1-ylmethyl)pyridine-3-carboxylic acid
3-(1-methylpiperidin-2-yl)-N-[1-(morpholin-4-ylmethyl)cyclohexyl]propanamide
2-methoxy-3-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
N-(furan-2-ylmethyl)-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidine-4-carboxamide
1-(3-{[({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)amino]methyl}phenyl)ethan-1-one
4-fluoro-3-({6-oxo-2,7-diazaspiro[4.5]decan-2-yl}sulfonyl)benzoic acid
(3S,4R)-1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-{1-[(3-methylphenyl)methyl]cyclopropyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
7-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,3-diazepane-2,4-dione
(3aR,6aS)-5-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{4-[(3-hydroxy-2,2-dimethylpropyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2,3-dimethoxy-N-{[1-(pyridin-3-ylmethyl)piperidin-3-yl]methyl}benzamide
N-[(3R,4S)-4-cyclopropyl-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-3-yl]cyclobutanecarboxamide
1-(5-chloropyridin-2-yl)-4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperazine
8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-[(2S)-5-oxopyrrolidine-2-carbonyl]-1,4-diazepan-2-one
5-{4-[2-(1,2-benzoxazol-3-yl)acetyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
5-acetyl-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N,2,4-trimethyl-1H-pyrrole-3-carboxamide
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
6-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}pyridin-3-ol
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-5-phenyl-1H-pyrrole-2-carboxamide
2-{4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrazine
(2-oxo-2-{7-[(pyridin-3-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}ethyl)urea
6-methoxy-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-{4-[(6-chloro-2-fluoro-3-methoxyphenyl)methyl]piperazin-1-yl}-1,3-thiazole-4-carboxamide
3-(5-methyl-1H-pyrazol-1-yl)-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]propanamide
1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)pent-4-en-1-one
(2S,4S)-N-ethyl-4-{4-[({[(3-methylphenyl)methyl]carbamoyl}amino)methyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-1-(4-hydroxypiperidin-1-yl)ethan-1-one
1-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
1-{4-[3-(1-benzothiophen-3-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperazin-1-yl}ethan-1-one
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
2-ethoxy-1-[4-(4-methoxybenzoyl)piperazin-1-yl]ethan-1-one
(3R,4R)-1-(2-methoxypyridine-4-carbonyl)-3,4-dimethylpyrrolidin-3-ol
2-methyl-5-[4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]pyrazine
2-(5-fluoro-2-methoxyphenyl)-N-(propan-2-yl)pyrimidin-4-amine
(4aR,7aS)-1-cyclopropanecarbonyl-4-(2-methoxypyrimidine-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-1H-indole
3-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]phenol
8-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
6-[4-(furan-2-carbonyl)-6-hydroxy-1,4-diazepan-1-yl]pyrazine-2-carboxamide