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[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl){[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
(3S,9aR)-3-benzyl-8-(4-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-(pyrrolidin-1-yl)pyridine-3-carboxamide
1-[1-(2,5-dimethoxybenzenesulfonyl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
dimethyl[3-(2-{1-[(2S)-pyrrolidine-2-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)propyl]amine
1-{1-[(5-phenylthiophen-2-yl)methyl]azetidin-3-yl}piperidine
N-[3-(morpholin-4-yl)propyl]-5-propyl-1,3,4-oxadiazol-2-amine
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
3-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2-fluoro-4-methylphenyl)-3-methylurea
5-{[methyl({5-[(5-methylfuran-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)amino]methyl}pyrimidin-2-amine
methyl 7-oxo-9-[2-(piperidin-1-yl)ethoxy]-3-(pyridine-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(4-ethylphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(3R,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-[3-(1H-imidazol-1-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(piperidin-1-ylmethyl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-1,4-oxazepane
4-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-oxazepane
5-methyl-N-{1-phenyl-3,6-diazatricyclo[4.3.1.13,8]undecan-9-yl}-1,3-oxazole-4-carboxamide
1-(4-methylphenyl)-3-{2-[4-(oxan-4-yl)morpholin-2-yl]ethyl}urea
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-[(2-methoxyethyl)(methyl)amino]propanamide
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
N'1-[4-(2,2-dimethylpropanamido)-3-methylphenyl]cyclopropane-1,1-dicarboxamide
6-methyl-2-oxo-5-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,2-dihydropyridine-3-carbonitrile
3-methyl-1-{2-oxo-2-[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethyl}-1,2-dihydroquinoxalin-2-one
2-[(2-aminopyridin-3-yl)methyl]-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3R,4R)-1-{2-[(dimethylcarbamoyl)amino]acetyl}-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
N-({3-methyl-7-[4-(thiophen-2-yl)butanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-phenylmethanesulfonamide
(1S,5R)-6-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-(azepan-1-yl)-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
(1S,5R)-6-methyl-3-[3-(4-phenylphenyl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4R)-N-ethyl-4-{[(3-fluorophenyl)methyl]amino}-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
3-(aminomethyl)-4-(4-tert-butylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{2-[({4-[1-(dimethylamino)ethyl]phenyl}methyl)(methyl)amino]ethyl}cyclopentan-1-ol
N-(3-chloro-4-methoxyphenyl)-3-{1-[2-(pyridin-2-yl)ethyl]piperidin-3-yl}propanamide
(1S,5R)-6-(2-methoxyethyl)-3-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]-6-(1H-pyrazol-1-yl)pyrimidine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(pyridin-3-yloxy)acetamide
3-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N4-methyl-N2-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}pyrimidine-2,4-diamine
3-(1H-imidazol-2-yl)-1-(3-phenoxybenzoyl)piperidine
8-[3-(ethylsulfanyl)propanoyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-6-methoxy-N-methylpyrimidin-4-amine
3-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-methylpyridazine
6-[5-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carbonyl]-1,2-dihydropyridin-2-one
5-({2-[3-(morpholin-4-yl)-3-oxopropyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(propan-2-yloxy)ethyl]acetamide
2-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
2-(1-ethylpiperidin-4-yl)-1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}ethan-1-one
1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(1H-pyrrole-2-carbonyl)piperazine