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1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
2-(3-chloro-4-hydroxyphenyl)-1-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}ethan-1-one
1-(2-phenylethyl)-3-(propan-2-yl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(6-ethoxyquinolin-2-yl)methyl](ethyl){[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
N4-methyl-N4-[2-(pyridin-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-6-(pyridin-4-yl)pyridine-3-carboxamide
(2E)-N-{[3-methyl-7-(1-methyl-1H-indole-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenylprop-2-enamide
5-(1-methyl-1H-pyrazol-4-yl)-4-phenyl-1-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-1H-imidazole
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(2-methoxyphenyl)propan-1-one
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(cyclopropylmethyl)acetamide
4-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-3-methyl-1-propyl-1H-pyrazole
1-[(4aS,7aR)-4-benzyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]cyclopropane-1-carboxamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
5-acetyl-6-methyl-3-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,2-dihydropyridin-2-one
2-[({5-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-4-(pyridin-4-yl)-1,4-diazepan-6-ol
methyl(oxolan-2-ylmethyl){[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
2-(quinolin-6-yl)pyridin-4-amine
2-(4-fluorophenyl)-N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
1-[2-(3-fluorophenyl)ethyl]-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-6-oxopiperidine-3-carboxamide
(1S,5R)-6-(4-methyl-1,3-thiazole-5-carbonyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(4aS,7aR)-1-(3-hydroxypyridine-2-carbonyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-cyclopentyl-2-(5-methoxyfuran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-(methylsulfanyl)propan-1-one
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidin-3-ol
4-[3-(3-chlorophenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,3-thiadiazole
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
3-methyl-7-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-3,4-dihydroquinazolin-4-one
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidine
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-3-methoxy-N-(oxolan-2-ylmethyl)benzamide
3-(2H-1,3-benzodioxol-5-yl)-1-(4-{2-[(2-methylphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)propan-1-one
6-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[1-(1-cyclopropylethyl)-3-methyl-1H-pyrazol-5-yl]-1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}urea
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[2-(propan-2-yl)-1H-1,3-benzodiazol-1-yl]ethan-1-one
1-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-2-(1H-imidazol-4-yl)-1H-imidazole
N2-[4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-N1-(pyridin-3-yl)ethane-1,2-diamine
{[2-(difluoromethoxy)phenyl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
2-(dimethylamino)-1-(4-methoxypiperidin-1-yl)-2-(2-methylphenyl)ethan-1-one
5-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(3aS,6aS)-2-(2-hydroxyethyl)-5-[(1-methyl-1H-indol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl](methyl){[3-(pyridin-2-ylmethoxy)phenyl]methyl}amine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-acetamido-2-methylpropanamide
4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine
5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidin-2-amine
2-({2-[(2-phenylethyl)(propyl)carbamoyl]phenyl}amino)acetic acid
(1S,4S)-2-({1-[1-(2-methylpyrimidin-4-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)-2-azabicyclo[2.2.1]heptane
2-(2,3-dihydro-1,4-benzodioxin-5-ylformamido)-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
4-[3-(4-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,6-dimethylpyrimidine
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(1,3-thiazol-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one