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1-tert-butyl-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-(3-{[(2-phenylpropyl)carbamoyl]methoxy}phenyl)propanamide
N-butyl-2-[methyl({4-oxo-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-6-yl})amino]acetamide
(1S,5R)-3-[5-(hydroxymethyl)furan-2-carbonyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[2-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)ethyl]-1-methylpiperidine
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-phenylbenzamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
5-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-N-benzyl-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-4-(morpholin-4-yl)butan-1-one
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(5-fluoro-2-methylbenzoyl)pyrrolidin-3-yl]methanol
4-(4-{[2-(2-hydroxyethyl)morpholin-4-yl]methyl}phenyl)-2-methylbutan-2-ol
N-(2,3-dihydro-1H-inden-2-yl)-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-2-(4-methoxyphenyl)pyrimidine
[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl})amine
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
N-cyclopentyl-3-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)propanamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-(pyridin-2-yl)ethan-1-one
(3S,5R)-1-(1-benzofuran-2-ylmethyl)-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
{5-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]furan-2-yl}methanol
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(1H-pyrazol-5-yl)benzamide
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-3-(1H-pyrazol-1-yl)propanamide
9-ethyl-1-methyl-4-(1,3-thiazol-4-ylmethyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-methyl-7-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(2-{4-[1-(4-methylpyridin-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)urea
(3R,5S)-1-benzyl-N-[(2,5-dimethylphenyl)methyl]-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
dimethyl[1-(3-{1-[2-(1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}phenyl)ethyl]amine
2-(1H-indazol-3-yl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}acetamide
(1R,5R)-6-(2-methoxyethyl)-N-(3-methylphenyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-methyl-N-[7-oxo-5-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]pentanamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(3,5-difluorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-ethyl-9-(1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-6-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-4-(1H-pyrazol-3-yl)benzamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamide
4-{2-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]ethyl}morpholine
1-[2-(methylsulfanyl)ethyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)morpholine
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-methoxypyrimidine
2-[2-(1H-imidazol-1-yl)ethyl]-1-{[4-(methylsulfanyl)phenyl]methyl}piperidine
8-(7-fluoro-2-methylquinoline-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-ethyl-1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
N-methyl-5-[(5-propylfuran-2-yl)methyl]-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-methoxy-2-phenyl-N-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
2-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}quinoline
4-{4-[(4-methoxyphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(ethylamino)pyridine-3-carboxamide
N-methyl-N-[2-(methylamino)ethyl]-3-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]benzene-1-sulfonamide
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-(2,5-dimethoxyphenyl)acetamide