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N-{[1-(adamantan-2-yl)piperidin-3-yl]methyl}-1-(4-chlorophenyl)cyclopropane-1-carboxamide
3-(3-fluorophenyl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1H-pyrazole-4-carboxamide
1-(2-methoxy-5-{[4-(3-methoxypropyl)piperidin-1-yl]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
1-ethyl-4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-cycloheptanecarbonyl-4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine
1-[2-(1H-pyrazol-1-yl)ethyl]-4-[3-(trifluoromethyl)phenoxy]piperidine
2-ethyl-N-[(8-methoxyquinolin-5-yl)methyl]-N-methylpyrimidine-5-carboxamide
7-({cyclopropyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-4-methyl-2H-chromen-2-one
2-(oxolan-2-ylmethyl)-9-(pyrazin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(1H-imidazol-1-yl)propyl]-1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
5-methyl-N-({3-methyl-7-[2-(2,3,6-trifluorophenyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)pyrazine-2-carboxamide
1-(3-chloropyridin-2-yl)-4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperazine
(1R,9aR)-1-[({3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
2-(4-{4-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)pyridine-3-carbonitrile
N-(propan-2-yl)-5-[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]pyrimidin-2-amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2,3-dihydro-1-benzothiophene-2-carboxamide
8-(1H-imidazol-4-ylmethyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
7-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{4-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]-3-methyl-1H-pyrazol-1-yl}ethan-1-ol
{1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-4-yl}(pyridin-2-yl)methanol
1-(3,4-dimethylphenyl)-N-(1,4-dithiepan-6-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-amino-6-(1-ethyl-1H-indol-3-yl)-4-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-[(4-chlorophenyl)methyl]-2-[(2S)-2-hydroxypropanoyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
8-[2-(2-hydroxyethoxy)ethyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-N-(2-methoxyethyl)cyclohexanecarboxamide
2-methoxy-1-[1'-(pyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-[(3-chlorophenyl)methyl]-2-methoxy-N-propylbutanamide
4-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-[2-(phenylsulfanyl)ethyl]-N-(prop-2-en-1-yl)-4-(4H-1,2,4-triazol-4-yl)benzamide
5-(3,5-dimethyl-1H-pyrrol-2-yl)-3-(oxolan-2-ylmethyl)-1,2,4-oxadiazole
3-methyl-1-propyl-4-[2-(thiophen-2-yl)azetidine-1-carbonyl]-1H-pyrazole
N-[1-(morpholin-4-ylmethyl)cyclopentyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
[(2-chloro-4-fluorophenyl)methyl]({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl})methylamine
methyl (1S,3S,3aR,6aS)-1-(hydroxymethyl)-5-methyl-3-(2-methyl-1-benzothiophen-3-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
4-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,3-dihydro-1H-imidazol-2-one
7-(3-chlorophenyl)-4-(6-methylpyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[1-(2,4-dimethylphenyl)propyl]-5-methyl-1,3,4-oxadiazole-2-carboxamide
2-(dimethylamino)-8-[3-methoxy-4-(prop-2-en-1-yloxy)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(furan-2-yl)-2-oxoacetamide
4-methoxy-N-(2-methoxyethyl)-2-{[1-(1,2-oxazole-3-carbonyl)piperidin-4-yl]oxy}benzamide
(3aS,6aS)-2-(5-ethyl-1,3,4-thiadiazol-2-yl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-ethyl-3-{1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoacetamide
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-(5-propyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]methanol
N-[(1S,2R)-2-aminocyclobutyl]-2-(1-oxo-4-phenyl-1,2-dihydrophthalazin-2-yl)acetamide
3-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-6-methylpyridazine
2-[3-oxo-9-(propane-2-sulfonyl)-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid