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(3S,9aR)-8-(2-fluorobenzenesulfonyl)-3-(1H-imidazol-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2-methyl-2-[4-(morpholin-4-yl)-2-[3-(pyridin-3-yl)azetidin-1-yl]pyrimidin-5-yl]propanoic acid
2-methyl-N-{2-oxo-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}propanamide
1-(3,4-dimethylphenyl)-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-N,N,5,6-tetramethylpyrimidin-2-amine
N-ethyl-2-{2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamido}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
5-({4-[3-(methoxymethyl)pyrrolidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}methyl)-1-methyl-1H-imidazole
{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
4-[(4-fluorophenyl)methyl]-1-(2-hydroxybenzoyl)-3-(propan-2-yl)-1,4-diazepan-5-one
5-[1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
1-[1-(3-cyano-6-methylpyridin-2-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
3-({4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carboxamide
3-[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-(furan-2-ylmethyl)propanamide
4-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-3-(4-fluorophenyl)-1H-pyrazole
1-[4-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)thiophen-2-yl]ethan-1-one
N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-2H-1,3-benzodioxole-5-carboxamide
3-butyl-4-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-1-methylpiperazin-2-one
2-methyl-5-(4-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
N-benzyl-4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-amine
(4aS,7aR)-1-[(2-chloro-4-fluorophenyl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
1-amino-N-butyl-N-[(4-fluorophenyl)methyl]cyclopropane-1-carboxamide
3-hydroxy-1-(2-methoxyethyl)-3-{[(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
(3S,7S)-5-(2-acetamidoacetyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
(2S,4S)-4-(2-hydroxy-4-methylbenzamido)-1-methylpyrrolidine-2-carboxylic acid
N-(1-benzyl-1H-pyrazol-3-yl)-2-[3-(3-fluorophenyl)-1H-pyrazol-1-yl]acetamide
7-(2-hydroxyethyl)-2-(2-phenylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
2-methoxy-N-methyl-5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)benzamide
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-7-fluoro-2-oxo-1,2-dihydroquinoline-4-carboxamide
4-(4-phenyl-1H-imidazole-5-carbonyl)-2-(trifluoromethyl)morpholine
3-cyclopropyl-1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
N-(2,2-difluoroethyl)-4-{[2-(pyridin-4-yl)ethyl]sulfamoyl}benzamide
4-[(4-fluorophenyl)methyl]-1-[2-(piperidin-1-yl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-(azocan-1-yl)-N-[(2-hydroxyphenyl)methyl]-N-methylpropanamide
dimethyl[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propyl]amine
3-methyl-4-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)piperazin-2-one
1'-(4-chlorobenzoyl)-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1R,9S)-5-amino-12-cyclopentyl-3-(1-ethyl-1H-pyrazol-4-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
(1R,5R)-6-[4-(1H-imidazol-1-yl)benzoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-cyclopropyl-3-{1-[4-(4-methoxyphenyl)-4-oxobutanoyl]piperidin-4-yl}propanamide
4-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-{1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]piperidin-4-yl}-N-(3-chloro-4-fluorophenyl)propanamide
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(quinolin-5-ylmethyl)acetamide
7-(cyclopropylmethyl)-2-[2-(2-methyl-1H-indol-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-methyl-5-(4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
methyl 6-benzyl-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-ethyl-3,5-dimethyl-N-(3-phenylprop-2-yn-1-yl)-N-propyl-1H-pyrazole-4-carboxamide
5-(3-{4-[(3,4-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}-3-oxopropyl)imidazolidine-2,4-dione