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(benzylsulfamoyl)(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)amine
N5-cyclooctyl-N3-(cyclopropylmethyl)-4-oxo-N3-propyl-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
1-[1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)azetidin-3-yl]-3,5-dimethyl-1H-pyrazole
N-(pyridin-3-ylmethyl)-3-(1H-1,2,4-triazol-3-yl)benzamide
(3R,4S)-4-cyclopropyl-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]pyrrolidin-3-amine
2-(1-cyclobutanecarbonylpyrrolidin-2-yl)-5-fluoro-1H-1,3-benzodiazole
2-(2H-1,3-benzodioxol-5-yl)-2-[methyl(pyridin-2-ylmethyl)amino]acetic acid
2-cyano-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]benzamide
(1,4-dioxan-2-ylmethyl)({[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl})methylamine
3-{[(1-ethylpyrrolidin-3-yl)carbamoyl]amino}-N-(2-methoxyethyl)-2-methylbenzamide
5-cyclobutanecarbonyl-1'-[(2S)-pyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(2,6-difluorophenyl)methyl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
5-[1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1H-1,2,3-triazol-4-yl]-2-(furan-2-yl)pyrimidine
2-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-1,2-dihydrophthalazin-1-one
{1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
3-[5-(phenoxymethyl)-1,3,4-oxadiazol-2-yl]-1-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
2-methoxy-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
1-[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-4-(1,3-thiazole-4-carbonyl)-1,4-diazepan-2-one
N-[(3R,4S)-4-cyclopropyl-1-(3,3-dimethylbutanoyl)pyrrolidin-3-yl]-2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-4-yl)acetamide
6-(3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)quinoxaline
4-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
1-ethyl-5-oxo-N-{[3-(trifluoromethoxy)phenyl]methyl}pyrrolidine-3-carboxamide
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
8-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{1-[6-(azepan-1-yl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
2-{4-[4-(1H-pyrazol-3-yl)benzoyl]piperazin-1-yl}pyrazine
4-{[(5-methylfuran-2-yl)methyl]amino}-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
(2E)-3-(1H-imidazol-4-yl)-1-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]prop-2-en-1-one
N-(furan-2-ylmethyl)-3-{[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]amino}propanamide
methyl({[1-(propan-2-yl)-1H-imidazol-5-yl]methyl})(quinolin-4-ylmethyl)amine
2-(dimethylamino)-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]benzamide
(2S)-2-amino-3-cyclohexyl-N-methyl-N-[2-(methylcarbamoyl)ethyl]propanamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-[methyl(piperidin-4-yl)amino]acetamide
4-[5-oxo-3-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-4-yl]benzoic acid
3-(2H-1,3-benzodioxol-5-yl)-5-(cyclopropylsulfamoyl)benzoic acid
1-(2-{methyl[(1-methyl-1H-indol-6-yl)methyl]amino}ethyl)cyclopentan-1-ol
7-(4-methanesulfonylphenyl)-1,2,3,4-tetrahydroisoquinoline
1-ethyl-5-methyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
4-{1-[4-(3-methoxyphenyl)phenyl]piperidin-4-yl}-1,2-dimethylpiperazine
1-({1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]cyclopropyl}methyl)-1H-pyrazole
methyl 8-(furan-3-ylmethyl)-1-(3-methylbutoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
3-[5-(3-methyl-1,2-oxazole-5-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
4-({2-[6-(piperazin-1-yl)pyridin-2-yl]phenyl}methyl)morpholine
3-{2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}imidazolidine-2,4-dione
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(propan-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-methyl-N-[2-methyl-2-(piperidin-1-yl)propyl]pyrimidin-2-amine
3-[(dimethylamino)methyl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-3-ol
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carboxamide