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(1S,5R)-3-[(4-fluorophenyl)methyl]-6-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
(2S,4R)-4-amino-1-[(2,2-difluoro-2H-1,3-benzodioxol-4-yl)methyl]-N-ethylpyrrolidine-2-carboxamide
2-{5-[(1S,2R)-2-(methylcarbamoyl)cyclohexyl]-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl}acetic acid
2-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-(adamantan-1-yl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-hydroxypyrimidine-5-carboxamide
2-(2-chloro-4-{[4-(oxan-4-yl)piperazin-1-yl]methyl}phenoxy)acetamide
3-(2-methoxyethyl)-1-[3-(4-methylphenyl)phenyl]-3-(oxolan-2-ylmethyl)urea
2-{1-[2-(3,5-difluorophenyl)ethyl]piperidin-2-yl}pyridine
1-{4-[4-(3-hydroxyphenyl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
N-cyclopropyl-3,3,3-trifluoro-2-hydroxy-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
2-(4-fluorophenyl)-2-[(2-propyl-1,3-thiazol-4-yl)formamido]acetic acid
1-[(2,3-difluorophenyl)methyl]-4-{1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]pyrrolidin-3-yl}piperidine
5-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-indole
1-[4-(difluoromethoxy)-2-methylphenyl]-3-ethyl-3-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]urea
4-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}-N-methylbenzene-1-sulfonamide
3-(6-methoxypyridin-3-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
1-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-(cyclopropylmethyl)-8-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N,N,2-trimethyl-7-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-cyclopentyl-3-(2-hydroxyphenyl)-3-(4-hydroxyphenyl)propanamide
2-methyl-4-{3-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]phenyl}butan-2-ol
2-[4-(5-tert-butyl-1H-pyrazol-3-yl)-1H-1,2,3-triazol-1-yl]-3-(furan-2-yl)propanoic acid
1-[(4-methoxyphenyl)methyl]-4-{thieno[2,3-d]pyrimidin-4-yl}piperazin-2-one
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(pyridin-4-yl)piperidin-4-yl]oxy}benzamide
2-[3-(2-methoxyphenyl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
1'-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}spiro[indene-1,4'-piperidine]
1-[7-(ethanesulfonyl)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]pyrrolidine
N-(1-propyl-1H-1,2,4-triazol-3-yl)-10-azabicyclo[4.3.1]decane-10-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}acetamide
(1R,3S)-7-(4-chloro-3-methylbenzoyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
5-[(3,4-dimethylpiperazin-1-yl)methyl]-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-cyclopropanecarbonyl-N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)piperidine-4-carboxamide
3-[4-(2-oxopyrrolidin-1-yl)piperidine-1-carbonyl]-1,2-dihydroquinoxalin-2-one
3-(1H-1,2,3-benzotriazol-4-yl)-1-[3-(cyclohexyloxy)propyl]urea
2-cyclopropyl-4-phenyl-9-(pyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecane
2-[2-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)ethoxy]ethan-1-ol
1-[2-(dimethylamino)ethyl]-N-methyl-6-oxo-N-{[2-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
2,2-dimethyl-3-[methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})amino]propan-1-ol
1-ethyl-N,2,5-trimethyl-N-(quinolin-5-ylmethyl)-1H-pyrrole-3-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
ethyl 2-(1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)acetate
3-[6-amino-5-cyano-4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)pyridin-2-yl]-1H-pyrazole-5-carboxylic acid
1-[1-(3-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}phenyl)ethyl]pyrrolidine
2,3-dimethyl-N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
(3R,9aR)-8-[(2-fluoro-5-methylphenyl)methyl]-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(2,3-dihydro-1H-inden-2-yl)-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
[(3R,4R)-4-(pyrrolidin-1-ylmethyl)-1-[4-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
4-(4-methylphenoxy)-N-[1-(thiophen-3-yl)propan-2-yl]piperidine-4-carboxamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide