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1-(2-cyclopropylacetyl)-4-[2-(1H-pyrazol-4-yl)ethyl]-1,4-diazepane-6-carboxylic acid
1-{4-[(1-methoxypropan-2-yl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
3-[(diethylcarbamoyl)methyl]-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-(3-chloro-5-fluorophenyl)-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1H-imidazole
methyl (1S,3S,3aR,6aS)-5-ethyl-3-(3-fluoro-5-methylphenyl)-1-(hydroxymethyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(1S,5R)-6-(2H-1,3-benzodioxol-5-ylmethyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-5,5-diphenylpiperidin-2-one
2-phenyl-8-(1H-1,2,3-triazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-1-one
5-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1-methyl-1H-1,2,3-benzotriazole
1-(2-chlorophenyl)-5-methyl-4-(1-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)piperazin-2-one
2-[(4aR,7aS)-4-[(2-methoxyphenyl)carbamoyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
3-[1-(3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
3-(2-methoxyethyl)-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylic acid
2-methyl-4-(1H-pyrazol-1-yl)-6-[3-(pyridin-2-yl)azetidin-1-yl]pyrimidine
{1-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
N-(1H-imidazol-2-ylmethyl)-7-methanesulfonyl-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1-(oxan-4-yl)piperidine-3-carboxamide
5-[4-(4-methylphenoxy)piperidine-1-carbonyl]-2-(pyridin-4-yl)pyrimidine
3-(3,5-dimethylphenyl)-N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}propanamide
2-cyclopentyl-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-phenylacetamide
2-(2-chlorophenyl)-3-methyl-N-[2-(1,3-thiazol-4-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
7-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-N-(prop-2-en-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-({5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)phenol
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-[1-(oxan-4-yl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-[4-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)morpholin-3-yl]-N-phenylacetamide
2-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-3-methoxyphenol
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
7-methoxy-5-{4-[1-(morpholin-4-yl)ethyl]phenyl}-1-benzofuran-2-carboxylic acid
(2R,6S)-4-[1-(2,3-difluoro-4-methoxybenzoyl)piperidin-4-yl]-2,6-dimethylmorpholine
2-{1-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]pyrrolidin-2-yl}pyridine
3-chloro-5-{4-oxo-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-1,2-dihydropyridin-2-one
1-{2-[({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]morpholin-4-yl}ethan-1-one
1-benzyl-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}piperidine-2-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
(2R,6R)-4-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-methyl-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrido[2,3-d]pyrimidin-4-amine
N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
3-(1-methyl-1H-imidazol-2-yl)-6-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}pyridazine
N-[(2R,4R,6S)-2-(4-chlorophenyl)-6-(isoquinolin-5-yl)oxan-4-yl]acetamide
2-(2-{2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]morpholin-4-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one
6-methyl-2-[1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
4-methyl-2-{1-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]propyl}pyridine
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(4-fluorophenyl)(pyridin-4-yl)methyl]propanamide
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-(2-methyl-1H-imidazol-1-yl)acetamide
2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)acetamide
(3S)-4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}pyridine-3-carboxylic acid
4-phenyl-N-{[1-(pyridin-4-yl)piperidin-3-yl]methyl}benzamide
1-(propan-2-yl)-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}piperidine-4-carboxamide
2-(3-chloro-4-hydroxyphenyl)-1-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]ethan-1-one