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N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1,9-dioxaspiro[5.5]undecan-4-amine
(1R,2s,3S,6R,7r,8S)-N-[3-(1H-imidazol-1-yl)propyl]-11,12-dioxatetracyclo[6.2.1.13,6.02,7]dodecane-2-carboxamide
N-[2-(2-fluorophenyl)-1-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)ethyl]-N,2-dimethylfuran-3-carboxamide
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}({[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
4-benzyl-3-butyl-1-[2-(3-methylpiperidin-1-yl)-2-oxoethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,5R)-6-benzyl-3-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-3,6-diazabicyclo[3.2.2]nonane
methyl 2-(N-methyl-1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazol-4-yl}formamido)acetate
1-{6-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]pyridin-2-yl}ethan-1-ol
(1R,5R)-N,N-dimethyl-6-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(3-chloro-4-methylphenyl)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}piperidin-4-amine
(1S,5R)-3-[3-(3-methoxyphenyl)propanoyl]-3,9-diazabicyclo[3.3.2]decan-10-one
[(1-ethylpyrrolidin-2-yl)methyl](furan-3-ylmethyl){[1-(2-methoxyethyl)piperidin-4-yl]methyl}amine
2-{5-[(3-oxo-2,3-dihydro-1H-isoindol-1-yl)methyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}acetic acid
4-[(4-fluorophenyl)methyl]-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3-(propan-2-yl)-1,4-diazepan-5-one
(3-{2-[1-(5-ethylthiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-N-methylpiperidine-2-carboxamide
1-{1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carbonyl}-1,4-diazepane
1,3-dimethyl-8-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(cyclohexylmethyl)-3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-methyl-2-(pyrrolidin-1-yl)propan-1-one
(cyclohex-3-en-1-ylmethyl)({[4-(3-methoxyphenyl)-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl})methylamine
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2-(4-ethylpiperazin-1-yl)ethan-1-one
3-({1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}methyl)-2,3-dihydro-1,3-benzoxazol-2-one
2-({[5-(1-benzoylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)ethan-1-ol
5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]pyrimidin-2-amine
3-{[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
2-ethyl-5-({4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidine
N-[2-(1H-imidazol-4-yl)ethyl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
2-{1-cyclohexyl-4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]-4-[(3-methylphenyl)methyl]piperazine
N-{2-methoxy-5-[2-(propan-2-yloxy)acetamido]phenyl}benzamide
N-(2,2-dimethylpropyl)-N-methyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(2S,4S)-4-amino-N-ethyl-1-{3-[(4-fluorophenyl)formamido]propanoyl}pyrrolidine-2-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1H-1,2,3-triazole-5-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-(5-fluoro-2-methylphenyl)acetamide
2-[2-(2-methoxyphenyl)ethyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-{1-[1-(methoxymethyl)cyclobutanecarbonyl]pyrrolidin-2-yl}-3,5-dimethyl-1,2-oxazole
[1-(morpholin-4-yl)propan-2-yl][(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
6-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-2-carbonitrile
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(1H-indol-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[4-(propan-2-yl)phenyl]-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
1-cyclopropanecarbonyl-3-[2-(3,4-difluorophenyl)ethyl]piperidine
4-(cyclopropylmethyl)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-ethyl-9-(1,2-oxazole-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,4R)-3-hydroxy-1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidin-4-yl]pyridine-4-carboxamide
3-[3-(3-chlorophenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrazine-2-carbonitrile
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-2-[3-(propoxymethyl)pyrrolidin-1-yl]pyrimidin-4-amine
[4-benzyl-1-(quinolin-2-ylmethyl)piperidin-4-yl]methanol