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2,6-dimethyl-5-{2-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-3,4-dimethyl-5-sulfamoylbenzamide
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
2-butoxy-1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
4-(3-hydroxy-3-methylbutyl)-N-[2-(1,3-thiazol-2-yl)ethyl]benzamide
4-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
5-ethyl-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-2-methylpyrimidin-4-amine
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-7-fluoro-2-methylquinoline-4-carboxamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 4-{[(1-cycloheptylpiperidin-3-yl)carbamoyl]amino}benzoate
1-[3-({[2-(furan-2-yl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
1-(1,4-dioxan-2-ylmethyl)-2-oxo-3-[2-(pyridin-2-yl)ethyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
(3R,4S)-4-{[(8-methoxyquinolin-2-yl)methyl](methyl)amino}oxolan-3-ol
1-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
N-(1H-indazol-4-yl)-4-[(3-oxopiperazin-1-yl)methyl]benzamide
1-cyclopropyl-4-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-(2-oxopyrrolidin-1-yl)benzamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}propane-1-sulfonamide
5-cyano-N,4-dimethyl-6-oxo-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,6-dihydropyridine-3-carboxamide
N-{1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}acetamide
5-{2-[1-(4-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]ethyl}imidazolidine-2,4-dione
4-hydroxy-2-[(3-phenylpiperidin-1-yl)methyl]quinoline-6-carboxamide
4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine-2-carboxylic acid
2-[(5-methylpyrazin-2-yl)methyl]-8-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-(dimethyl-1,2-oxazol-4-yl)-1-(2-phenylethyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(2-methyl-4-oxopentanoyl)piperidin-4-yl]oxy}benzamide
N-(3-methoxypropyl)-4-methyl-N-(1-methylpiperidin-4-yl)-1,3-oxazole-5-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
N-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]pyrazolo[1,5-a]pyridine-7-carboxamide
4-({4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepan-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
{2-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}urea
6,7-dimethoxy-2-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
3-{1-[1-(propan-2-yl)piperidine-4-carbonyl]azetidin-3-yl}pyridine
3-{1-[2-(pyridin-4-yl)ethyl]-1H-imidazol-2-yl}quinolin-7-ol
2-(2,2-dimethylpropanoyl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-(3-hydroxybenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-[2-(2-phenylethyl)morpholin-4-yl]acetic acid
methyl 2-{2-[(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamido)methyl]-5-methyl-2,3-dihydro-1-benzofuran-7-yl}benzoate
(4aR,8aS)-1-[2-(4-methoxyphenyl)ethyl]-6-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-decahydro-1,6-naphthyridin-2-one
1-(cyclobutylmethyl)-3-hydroxy-3-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]piperidin-2-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[2-(3-fluorophenyl)ethyl]-N-methyl-6-oxopiperidine-3-carboxamide
N-methyl-N-(1H-pyrazol-3-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-({8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)benzonitrile
4-[3-(morpholin-4-yl)azetidine-1-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-({[(4-methylphenyl)methyl]amino}methyl)piperidin-2-one
1-tert-butyl-4-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrrolidin-2-one
5-(methoxymethyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,3,4-oxadiazole-2-carboxamide
(3R,5S)-N3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N5-(4-methylphenyl)piperidine-3,5-dicarboxamide
2-methyl-4-(4-{[(1r,5r)-7,10-dimethyl-3,7,10-triazatricyclo[3.3.3.01,5]undecan-3-yl]methyl}phenyl)butan-2-ol
5-cyclobutanecarbonyl-1'-(1H-imidazol-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]