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1-(4-methoxybenzoyl)-4-(4-methyl-1,3-thiazole-5-carbonyl)piperazine
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[(4-sulfamoylphenyl)methyl]propanamide
N-methyl-6-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
[(3R,4R)-1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[3-(3-chlorophenyl)phenyl]-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
2-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1,4-diazepan-6-yl)acetic acid
5-cyclobutanecarbonyl-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-3-(2-methyl-1H-1,3-benzodiazol-6-yl)urea
5-tert-butyl-4-({5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}methyl)furan-2-carboxamide
5-{2-[2-(propylamino)pyrimidin-5-yl]-1H-imidazol-1-yl}pyridine-3-carboxylic acid
(1S,9R)-11-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-(1-benzothiophen-7-yl)-2-(4-hydroxypiperidin-1-yl)acetic acid
4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-2-chlorobenzoic acid
1-{1-[(3-methoxyphenyl)methyl]-5-(thiophen-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
1-(2-fluoro-5-methanesulfonamidophenyl)-3-(pentan-2-yl)urea
6-fluoro-2-{[4-(propan-2-yl)piperazin-1-yl]methyl}quinolin-4-ol
3-ethyl-5-hydroxy-N-{2-[(pyridin-3-yl)amino]ethyl}adamantane-1-carboxamide
4-(1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)thiomorpholine
2-[(prop-2-en-1-yl)amino]-N-{3-[(pyridin-3-yl)amino]propyl}benzamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidine
N-[(5-{[(1s,4s)-4-aminocyclohexyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
3-[methyl(pyrazin-2-ylmethyl)sulfamoyl]-N-(pyridin-3-yl)benzamide
4-[2-(5-methyl-1H-pyrazol-1-yl)ethyl]-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]ethan-1-one
N-(2-hydroxyethyl)-2-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-benzofuran-7-carboxamide
6-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,3-benzothiazole
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-(oxolan-3-ylmethyl)pyrimidine-5-carboxamide
2-(2-hydroxyethyl)-9-[2-(4-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
1-benzyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H-pyrazole-4-carboxamide
(2R,3S,6R)-5-(2-fluorobenzoyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-[(4-methoxypyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-{1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-imidazol-2-yl}-4,5,6,7-tetrahydro-1,3-benzothiazole
1-benzyl-8-{[4-(furan-2-yl)phenyl]methyl}-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(5-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}thiophen-3-yl)methyl]dimethylamine
3-(4-methoxyphenyl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1H-pyrazole-5-carboxamide
5-(piperidin-4-yl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
4-(6-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrazine-2-carbonyl)morpholine
(3R,4R)-4-(azepan-1-yl)-1-[1-(2-methoxyphenyl)piperidin-4-yl]piperidin-3-ol
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(methylamino)-1,3-thiazole-4-carboxamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-[2-(1H-pyrazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
(3S,4S)-1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-{3-hydroxy-1-[4-(propan-2-yl)phenyl]propyl}-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
2-[2-fluoro-3-(trifluoromethyl)phenyl]-6-(pyrrolidine-1-carbonyl)pyrazine
1-[(2R,3R)-3-[ethyl(methyl)amino]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(pyrrolidin-1-yl)ethan-1-one
2-[3-methyl-4-({4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}methyl)-1H-pyrazol-1-yl]ethan-1-ol
(4aS,7aR)-1-{imidazo[1,2-a]pyridine-3-carbonyl}-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,6-dimethyl-4-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)phenyl acetate
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide