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1-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
2-[4-chloro-2-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]acetamide
1-[3-(morpholin-4-yl)propyl]-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]piperidin-2-one
4-methyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)piperidine-1-sulfonamide
(3S,4R)-N,N-dimethyl-1-[(6-methylpyridin-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-amine
N-{[(2R)-1-ethylpyrrolidin-2-yl]methyl}-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
7-methyl-2-[2-(morpholin-4-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
3-methyl-6-[5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]pyridazine
[(2S,6S)-4-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]butan-1-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-(pyridin-4-ylsulfanyl)acetamide
N-ethyl-4-methyl-5-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]-1,3-thiazol-2-amine
1-[2-(3-methoxyphenyl)piperidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
3-(1H-imidazol-4-ylmethyl)-4-{2-[1-(propan-2-yl)piperidin-4-yl]acetyl}piperazin-2-one
(1R,5R)-N,N-dimethyl-6-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-3-phenylpropanamide
2-[3-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)phenyl]-5-methyl-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
5-ethyl-N4-[(1S)-1-(3-methylpyridin-2-yl)ethyl]pyrimidine-2,4-diamine
N-[(4-chlorophenyl)methyl]-3-[4-(4-cyanophenyl)-3-oxopiperazin-1-yl]propanamide
3-ethyl-N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-5-methyl-1,2-oxazole-4-carboxamide
1-(cyclopropylmethyl)-5-[5-(methoxymethyl)thiophene-2-carbonyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]propan-1-one
1-(2-methoxyethyl)-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-6-oxopiperidine-3-carboxamide
(2S,4S)-4-amino-1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[(4-methoxyphenyl)methyl]-N-[1-(thiophen-3-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
10-methoxy-5-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N,5-dimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-[(3-phenylpropyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
(3R,4S)-4-cyclopropyl-1-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-amine
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-(2,4,6-trimethylphenoxy)ethyl]propanamide
2-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3-hydroxypyrrolidin-3-yl)methyl]quinoline-6-carboxamide
1-(3-chloro-4-methoxyphenyl)-5-oxo-N-[2-(pyridin-3-yl)ethyl]pyrrolidine-3-carboxamide
2-cyclohexyl-1-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-4-(2,4-dioxoimidazolidin-1-yl)benzamide
1-[1-(5-methoxypyridin-3-yl)-3,5-dimethyl-1H-pyrazol-4-yl]propan-2-one
N-[2-(3-fluorophenyl)ethyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
5-(3-chlorophenyl)-3-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-1,2,4-triazine
3-[5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]benzonitrile
1-[2-(azepan-1-yl)ethyl]-4-ethyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(3-hydroxy-3-methylbutyl)-N-[1-(4-hydroxyphenyl)ethyl]benzamide
(3R,4R)-4-amino-1-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]piperidin-3-ol
1-(cyclohex-3-en-1-ylmethyl)-4-[(2,6-dimethylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
5-{1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-1H-imidazol-2-yl}-2-(pyridin-2-yl)pyrimidine
N-{[3-(2-chlorophenyl)phenyl]methyl}acetamide
3-(azepane-1-carbonyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3,4-difluoro-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]benzamide
1,3-dimethyl-2,6-dioxo-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[7-oxo-5-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]thiophene-3-carboxamide