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dimethyl(3-{2-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
N-[4-({[(3-methoxyphenyl)methyl](prop-2-en-1-yl)amino}methyl)phenyl]acetamide
2,5-dimethyl-N-[(1S,2R)-2-{[1-(propan-2-yl)piperidin-4-yl]amino}cyclobutyl]thiophene-3-sulfonamide
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
1-{1-[(6-chloropyridin-3-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
ethyl 4-(3-{[(4-phenylphenyl)formamido]methyl}piperidin-1-yl)piperidine-1-carboxylate
8-(2-butoxyacetyl)-2,8-diazaspiro[4.5]decan-3-one
2-[5-cyclopropyl-4-(4-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]-4-(3-fluoro-4-methoxyphenyl)pyrimidine
5-fluoro-6-methyl-2-{4-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
2-(5-acetylthiophen-3-yl)-N-({4-[(dimethylamino)methyl]phenyl}methyl)acetamide
methyl({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amine
3-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-1-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-4-(furan-2-ylmethyl)-1,4-diazepan-6-ol
1-[(1-benzyl-1H-imidazol-2-yl)methyl]-4-ethyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1-{[methyl({[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl})amino]methyl}cyclopropyl)methanol
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1-(5-propylpyrimidin-4-yl)piperidin-4-amine
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-(propane-2-sulfonyl)piperidine
N-tert-butyl-4-(1-methyl-1H-1,2,3,4-tetrazol-5-yl)benzene-1-sulfonamide
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
(2S,4R)-1-[(3-chlorophenyl)methyl]-N,N-diethyl-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
6-({[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
7-fluoro-2-methyl-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]quinoline-4-carboxamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
3-({2-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
N-cyclohexyl-3-{[4-hydroxy-2-(pyridin-2-yl)pyrimidin-5-yl]formamido}propanamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)acetamide
N-methyl-5-[3-(1-methylpiperidin-2-yl)propanoyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N,4-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-(2-oxoimidazolidin-1-yl)benzamide
5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-[2-(5-methylfuran-2-yl)propyl]-1H-1,2,3-triazole
(2S,4R)-N,N-diethyl-1-(2-hydroxybenzoyl)-4-(2-methoxyacetamido)pyrrolidine-2-carboxamide
5-{[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
4-(4-{1-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
2-ethyl-8-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3,5-dimethyladamantane-1-carboxamide
2-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-6-methoxyphenol
3-(2-chlorophenyl)-N-cyclopropyl-3-phenylpropanamide
3-(4-methanesulfonylphenyl)-5-(2-methylpropyl)-1H-1,2,4-triazole
8-(2,4,5-trifluorobenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[2-(dimethylamino)ethyl]-4-[4-(2-methoxyacetyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
N-(1-{1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
7-(cyclohexylmethyl)-2-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-1-methylcyclopropane-1-carboxamide
N-(4-fluorophenyl)-1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidin-3-amine
N-(2-oxoazepan-3-yl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[1-(pyrimidin-4-yl)ethyl]acetamide