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4-chloro-1-ethyl-N-[2-(1H-imidazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
(3S,4S)-4-cyclopropyl-1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)pyrrolidine-3-carboxylic acid
(1S,5R)-6-(2,6-dimethylpyrimidine-4-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
6-methyl-2-(1-methyl-1H-pyrazol-4-yl)-4-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]quinoline
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-3,3-diphenylpiperidine
({6-[(3-fluorophenyl)methoxy]-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
(1R,5R)-N,N-dimethyl-6-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-[(4-methylpiperidin-1-yl)methyl]piperidin-2-one
5-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-{[3-(2-methylphenyl)phenyl]methyl}piperidine
1-[(4aR,8aR)-7-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
2-amino-4-[2-(2-hydroxyethoxy)phenyl]-6-(2-methylbutan-2-yl)pyridine-3-carbonitrile
2-(cyclopent-2-en-1-yl)-1-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]ethan-1-one
4-[4-(4-methylphenyl)-2-{[1-(pyrimidin-4-yl)ethyl]amino}pyrimidin-5-yl]phenol
N-[(2R)-pyrrolidin-2-ylmethyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
6-methyl-5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[4-(4-chlorophenyl)piperazin-1-yl]-3-(3-methylpiperidin-1-yl)propan-1-one
1-[4-(2-fluorophenyl)benzoyl]-4-methyl-1,4-diazepan-5-one
N-cyclopentyl-3-fluoro-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}benzamide
1-[2-(4-methyl-1H-pyrazol-1-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-(propan-2-yl)piperidine-4-carboxamide
2-methyl-6-[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl]pyrimidin-4-ol
1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-3-(1-methyl-1H-pyrrol-2-yl)propan-1-one
N-methyl-N-{[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3-[4-(methylsulfanyl)benzoyl]piperidine
3-(1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}azetidin-3-yl)pyridine
4-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]pyrrolidin-2-yl}-3,5-dimethyl-1,2-oxazole
N-{[(3S,4S)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-hydroxypiperidin-4-yl]methyl}pyrrolidine-1-carboxamide
N-(oxolan-2-ylmethyl)-2-(1,3-thiazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(3-methylthiophen-2-yl)-1H-imidazole
methyl({[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
(2R,6S)-2,6-dimethyl-4-({3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)morpholine
4-methyl-N-{2-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-(1,2-diphenylethyl)-3-(2-ethyl-5-oxopyrrolidin-2-yl)propanamide
N-[2-(2-chlorophenyl)ethyl]-3-(1-methylpiperidin-4-yl)propanamide
1,3-dimethyl-N-(oxan-3-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-[3-(dimethylamino)propyl]-1-(2-phenylethyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-ethoxy-4-({[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amino}methyl)phenol
3-[2-(4-fluorophenyl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
N-(3,3-diphenylpropyl)-6-[2-(1H-imidazol-1-yl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(2-hydroxyethyl)acetamide
3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]propanamide
4-{[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]methyl}-1-ethyl-1H-pyrrole-2-carbonitrile
N-(4-{[1-(2-methoxyethyl)-2,4-dioxo-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}phenyl)acetamide
2-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-2-(dimethyl-1,2-oxazol-4-yl)acetic acid
3-benzyl-1-methyl-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,3-dimethyl-2-oxo-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-2,3-dihydro-1,3-benzoxazole-5-carboxamide