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5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[2-(pyrazin-2-yl)ethyl]-1H-pyrazole-3-carboxamide
1-(cyclohexylmethyl)-5-[(2-hydroxyethyl)(methyl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3R,4R)-1-(2-methoxy-4-methylbenzoyl)-3,4-dimethylpyrrolidin-3-ol
N,N-dimethyl-5-{2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetyl}-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
4-{[5-(2-methyl-1-benzothiophen-3-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
N-tert-butyl-2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetamide
1-ethyl-3,5-dimethyl-4-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}-1H-pyrazole
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethan-1-one
5-phenyl-N-(2,2,2-trifluoroethyl)pyrazolo[1,5-a]pyrimidin-7-amine
3-{[(6-fluoro-4-hydroxyquinolin-2-yl)methyl](methyl)amino}-N-methylbutanamide
{5-[4-(thian-4-yl)piperazine-1-carbonyl]-1H-1,3-benzodiazol-2-yl}methanol
(4aS,8aR)-6-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
N-cyclopentyl-3-{[(4-fluorophenyl)methyl]amino}-5-(phenylsulfamoyl)benzamide
1-[1-(2-aminoacetyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-4-carboxamide
3-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-ol
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(2-methylpyridin-4-yl)methyl]pyridin-2-amine
2-[3-(1H-pyrazol-1-yl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(1H-pyrazol-1-ylmethyl)benzamide
2-(4-{[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}phenoxy)pyrimidine
(1R,7S)-3-(2-ethylbutyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-[2-(3,4-dimethoxyphenyl)ethyl]-4-{4-[2-(4-methylphenoxy)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
(3S,4R)-N,N-dimethyl-4-propyl-1-{[5-(1H-pyrazol-5-yl)furan-2-yl]sulfonyl}pyrrolidin-3-amine
1-[(3S)-3-ethylmorpholin-4-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N,N-dimethylpiperidine-1-carboxamide
4,6-dimethyl-3-[4-(thian-4-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
(2R,3R)-3-amino-1'-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[(4-chlorophenyl)methyl]-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-6-oxopiperidine-3-carboxamide
3-[1-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-7-fluoro-3,4-dihydroquinazolin-4-one
2-(2-chlorophenyl)-N-[(1-ethyl-1H-imidazol-5-yl)methyl]-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
methyl 2-[3-(propan-2-yl)-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]acetate
N-(2,2-difluoroethyl)-4-(3-ethyl-3-hydroxypiperidine-1-carbonyl)benzene-1-sulfonamide
5-(3-propyl-1,2,4-oxadiazol-5-yl)-1-(pyridin-2-ylmethyl)piperidin-2-one
2-butyl-8-(2-hydroxy-3-methoxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-4-[(2-hydroxyethyl)sulfamoyl]benzamide
N,8-dimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-(3-chloro-4-fluorophenyl)-2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carboxamide
3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}urea
5-{imidazo[1,2-a]pyridine-2-carbonyl}-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[4-({3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
3-[2-(3-chlorophenyl)-1H-imidazol-1-yl]pyridin-2-ol
2-(2H-1,3-benzodioxol-5-yl)-N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
(3S,4S)-1-[methyl(propan-2-yl)sulfamoyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
(2S,4S,5R)-5-(4-chlorophenyl)-1,2-dimethyl-4-(morpholine-4-carbonyl)pyrrolidine-2-carboxylic acid
N-[4-(2-chlorophenyl)-2-methoxyphenyl]acetamide
2-hydroxy-N-[(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}pyrrolidin-3-yl)methyl]acetamide
(2S,4S)-4-amino-1-[2-(ethylamino)pyrimidine-5-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-(oxolane-2-carbonyl)-1-(2-phenylethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
methyl 4-[5-({[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate