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4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-cyclopentylpiperazin-2-one
5-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole
N-cyclopropyl-1-{1-[2-(4-fluorophenyl)acetyl]piperidin-4-yl}piperidine-4-carboxamide
5-{[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[2-(3-fluorophenyl)ethyl]-2-[4-(4-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}piperidin-1-yl)phenyl]acetamide
4-[2-(2-aminoethyl)quinazolin-4-yl]-3-methyl-1-[(3-methylphenyl)methyl]piperazin-2-one
(3aS,6aS)-2-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[5-cyclopropyl-4-(4-methylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(3-fluoro-4-methoxyphenyl)pyrimidine
3-{2-[4-(dimethylamino)azepan-1-yl]-2-oxoethyl}-5-methyl-2,3-dihydro-1,3-benzoxazol-2-one
1-(4-{4-[2-(hydroxymethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)-3-methoxypropan-1-one
methyl 2-[(2,3-dihydro-1H-inden-5-yl)sulfamoyl]-6-(2-ethylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(2S,4S)-N-ethyl-4-(3-methoxybenzamido)-1-(3-methoxypropanoyl)pyrrolidine-2-carboxamide
3-(1-methylpiperidin-2-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-8-azabicyclo[3.2.1]octane
N-{3-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-3-oxopropyl}acetamide
N-benzyl-5-[(2,6-difluorophenyl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2-methoxyethyl)-6-oxo-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}piperidine-3-carboxamide
2-(4-methoxyphenyl)-N-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methyl]acetamide
2-[3-(dimethyl-1,3-thiazol-5-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2,2-bis(prop-2-en-1-yl)piperidine
(4aS,7aR)-1-(4-hydroxy-3-methoxybenzoyl)-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3-phenylpyrrolidin-3-ol
2,3-difluoro-N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]benzamide
2-{[4-(2,4,6-trimethylphenyl)phenyl]methoxy}ethan-1-amine
2-{2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
N-(1,3-dihydroxypropan-2-yl)-2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]acetamide
4-fluoro-N-[3-(2-methyl-5-oxo-1,4-diazepan-1-yl)-3-oxopropyl]benzamide
3-(1-methyl-1H-pyrazol-5-yl)-N-[2-(pyrrolidin-1-yl)ethyl]propanamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N-methylpyrimidin-4-amine
5-methyl-4-[(4-methyl-1H-pyrazol-1-yl)methyl]-2-[4-(methylsulfanyl)phenyl]-1,3-oxazole
11-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-4-carbonitrile
3-(5-methyl-1,2,4-oxadiazol-3-yl)-N-(6-phenoxypyridin-3-yl)piperidine-1-carboxamide
4-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-2-methoxyphenol
2-(azepan-1-yl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
8-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-1-oxa-8-azaspiro[4.5]decane
4-{[1-(2-ethylpyridine-4-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamide
8-(3-methylbenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-cyclopentanecarbonyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}piperidine-4-carboxamide
3-(dimethyl-1H-1,2,4-triazol-1-yl)-N,2-dimethyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
8-fluoro-2-({[(1r,4r)-4-hydroxycyclohexyl]amino}methyl)quinolin-4-ol
N-[(2,6-dimethoxyphenyl)methyl]-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
N-(2-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)methanesulfonamide
(3S,9R)-11-(4-phenylbenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
8-fluoro-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}quinoline-2-carboxamide
2-(2-methoxyphenoxy)-N-{[1-(1H-pyrazole-4-carbonyl)piperidin-3-yl]methyl}acetamide
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl})amine