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N-{3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}naphthalene-1-sulfonamide
2-(cyclohex-1-ene-1-carbonyl)-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-methylpiperidin-2-one
N-(3-methoxyphenyl)-3-[1-(oxane-2-carbonyl)piperidin-4-yl]propanamide
1-ethyl-4-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-5-methyl-1H-pyrazole
3-{5-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-ylmethyl]thiophen-3-yl}prop-2-yn-1-ol
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]oxane-4-carboxamide
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-hydroxy-2-phenylpropan-1-one
N-[(5-oxopyrrolidin-2-yl)methyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
N-ethyl-1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]pyrrolidine-3-carboxamide
2-(2,4-dichlorophenoxy)-1-[2-(ethoxymethyl)pyrrolidin-1-yl]ethan-1-one
5-cyclopentanecarbonyl-3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(5-methyl-1H-pyrazol-1-yl)propanamide
(2S,4R)-N-[2-(4-fluorophenyl)ethyl]-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
N-[4-({[2-(pyridin-2-yl)ethyl]carbamoyl}methyl)phenyl]butanamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(1H-pyrazol-3-yl)benzamide
9-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
2-cyclopropyl-6-oxo-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]-1,6-dihydropyrimidine-5-carboxamide
1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3-[(dimethylamino)methyl]pyrrolidin-3-ol
4-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
{4-[4-(1H-pyrazol-1-yl)phenyl]pyridin-2-yl}methanol
N-[2-(azepan-1-yl)ethyl]-N-ethyl-2,6-dimethoxypyridine-3-carboxamide
5-tert-butyl-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1,3,4-oxadiazol-2-amine
4-[1-(2-methoxyacetyl)piperidin-3-yl]benzoic acid
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-5-methylpiperidin-2-one
4-[(2-fluoro-4-methoxyphenyl)methyl]-2-(2-methoxyethyl)morpholine
1-[2-(ethanesulfonyl)ethyl]-5,5-diphenylpiperidin-2-one
1-(2-{[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]methyl}-5-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
6-[1-(1-benzothiophene-2-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]pyrazolo[1,5-a]pyridine-3-carboxamide
N-({5-[3-(dimethylamino)-2,2-dimethylpropyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
2-amino-4-[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]-6-(3,4,5-trifluorophenyl)pyridine-3-carbonitrile
(3S,4S)-1-(3-ethyl-1H-pyrazole-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
(2S,4S)-4-amino-1-[2-amino-6-(2-methylpropyl)pyrimidine-4-carbonyl]-N-ethylpyrrolidine-2-carboxamide
1-[2-({3-azaspiro[5.5]undecan-9-yl}amino)ethyl]imidazolidin-2-one
5-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-3-methyl-1H-1,2,4-triazole
4-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)piperazine-2-carboxylic acid
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-3-(1H-pyrazol-1-yl)benzamide
1-{4-methyl-2-[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]pyrimidin-5-yl}ethan-1-one
3-chloro-5-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
1-(8-fluoroquinoline-2-carbonyl)-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
2-benzyl-9-(5-ethyl-2-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-{[5-(2-phenyl-1,3-thiazol-5-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
N-(2-{4-[(6-methylpyridin-2-yl)methyl]morpholin-2-yl}ethyl)cyclopropanesulfonamide
({5-[1-(1H-1,3-benzodiazole-5-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
{4-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]phenyl}methanol
2-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one