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N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1,2-oxazinan-2-yl)propanamide
2-(dimethyl-1,2-oxazol-4-yl)-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)acetamide
N-[(2,3-difluorophenyl)methyl]-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl][(3-{[1-(pyridine-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
4-[2-(1-{[2-(methylsulfanyl)phenyl]methyl}piperidin-2-yl)ethyl]morpholine
2-(4-chlorophenyl)-4-[(4,6-dimethylpyrimidin-2-yl)methyl]morpholine
3-(4-ethyl-1H-pyrazol-5-yl)-1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidine
4-benzyl-3-ethyl-1-[2-(pyrrolidin-1-yl)acetyl]-1,4-diazepan-5-one
[1-(4-ethenylbenzoyl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(3-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
(2S,4S,5R)-1-methyl-4-(4-methyl-1,4-diazepane-1-carbonyl)-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
2-[(3S)-3-ethylmorpholine-4-carbonyl]-5-methoxy-4H-pyran-4-one
3-(1H-indol-3-yl)-N-({8-[(2-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)propanamide
N,N-dimethyl-3-[({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amino)methyl]pyridin-2-amine
[(3R,4R)-1-{[4-(methylsulfanyl)phenyl]methyl}-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-(3-fluorophenyl)-4-(5-methyl-2-phenylfuran-3-carbonyl)piperazin-2-one
2-methyl-6-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)-2,3-dihydropyridazin-3-one
6-ethoxy-3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
2-phenyl-5-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
1-(6-fluoro-4-methylquinazolin-2-yl)-N-[2-(2-fluorophenyl)ethyl]azepan-4-amine
2-[3-(pyridin-3-yl)azetidine-1-carbonyl]-1,4-dihydroquinolin-4-one
4-{4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]phenoxy}-N,N-dimethylpiperidine-1-sulfonamide
1-acetyl-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)piperidine-4-carboxamide
N-(4-fluoro-2-methylphenyl)-3-[1-(1,3-thiazol-5-ylmethyl)piperidin-3-yl]propanamide
4-ethyl-3-[1-(9H-purin-6-yl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,5S)-N-(4-fluorophenyl)-1-(2-methylpropyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
9-[2-(2,3-difluorophenyl)acetyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carbonyl]-5-methoxy-1,4-dihydropyridin-4-one
N,N,2-trimethyl-7-(3-phenyl-1H-pyrazole-5-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(4-fluorophenoxymethyl)-4-hydroxy-N-methyl-N-(1-methylpyrrolidin-3-yl)pyrimidine-5-carboxamide
2-(methylsulfanyl)-6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
1-methyl-2-[1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
2-[3-(dimethylamino)propyl]-9-(2-ethylpyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethyl]methanesulfonamide
methyl 5-(2,2-dimethyloxane-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-cyclobutanecarbonyl-N-[3-(2-fluorophenyl)propyl]piperidine-4-carboxamide
2-methyl-8-[4-(5-methylfuran-2-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
2-methyl-4-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,3-thiazole
2-{2-[1-(quinoxaline-6-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N2-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyrimidine-2,4-diamine
{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(2-methyl-1H-indol-1-yl)ethyl]acetamide
4-[1-benzyl-5-(thiolan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
N-cyclohexyl-3-{methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}propanamide
5-[(3-chlorophenyl)methyl]-7-oxo-2-(pyrrolidin-1-yl)-4H,7H-pyrazolo[1,5-a]pyrimidine-3-carbonitrile
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-3,5-dimethylfuran-2-carboxamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-(4-phenylazepan-1-yl)ethan-1-one
2-(6-fluoroquinolin-8-yl)-4,5,6-trimethylpyridine-3-carbonitrile
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide