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1-(propan-2-yl)-4-{4-[3-(propan-2-yloxy)phenyl]-1H-imidazol-2-yl}pyrrolidin-2-one
N-[(5-chlorothiophen-2-yl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-(propan-2-yl)-9-(1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(3S)-3-ethyl-4-[4-(1-phenyl-1H-imidazol-4-yl)benzoyl]morpholine
5-[1-(2,4-difluoro-3-methoxybenzoyl)pyrrolidin-2-yl]thiophene-2-carboxamide
1-ethyl-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-{[1-(propan-2-yl)cyclopropyl]carbamoyl}pyrrolidine-2-carboxylic acid
4-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)benzonitrile
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-phenylazepane
N-[2-(2-methoxyphenyl)ethyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
8-methyl-3-({methyl[(3-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-[(3S,4R)-1-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(2,4-dimethoxy-3-methylphenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
methyl 2-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]sulfonyl}-6-[(2,5-dimethylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(1S,4R)-2-{[2-(trifluoromethyl)phenyl]methyl}-2-azabicyclo[2.2.1]heptan-3-one
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
4-[1-(3-chlorophenyl)-1H-pyrazol-4-yl]-N-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]pyrimidin-2-amine
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-imidazole-2-carboxamide
3-[5-(2,3-dihydro-1H-indene-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
3-(morpholine-4-carbonyl)-1-propyl-N-{[3-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
2,5-dimethyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]furan-3-carboxamide
2-(dimethylamino)-2-(2-methylphenyl)-1-[3-(morpholin-4-yl)azetidin-1-yl]ethan-1-one
1-cyclopentyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N-[(2-methoxyphenyl)methyl]-N-[(3-methylphenyl)methyl]-2-(5-oxopyrrolidin-2-yl)acetamide
(3R,4S)-1-[2-chloro-5-(trifluoromethyl)benzoyl]-4-propylpyrrolidin-3-amine
methyl 4-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}benzoate
7-(3-chlorophenyl)-9-[(1-methylpiperidin-3-yl)methoxy]-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{2-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]phenyl}-N-methylpropanamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-methyl-9-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
4-(4-{1-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
4-(benzyloxy)-1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
2-(3-methoxyphenyl)-1-{pyrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidine
4,4,4-trifluoro-N-[(4-methoxyphenyl)methyl]-N-(2-methylpropyl)butanamide
3-[5-({4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)-1,3,4-oxadiazol-2-yl]pyridine
1-(3-{[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenyl)ethan-1-one
2-[(3-phenoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane
7-(3-methoxyphenyl)-2-[1-(propan-2-yl)-1H-imidazol-2-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[(3,4-dimethylphenyl)amino]-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]cyclohexane-1-carboxamide
6-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carbonitrile
N-{[6-(6-methylquinolin-5-yl)pyridin-3-yl]methyl}acetamide
6-(4-methoxyphenyl)-7-methyl-8-oxo-N-[(2R)-pyrrolidin-2-ylmethyl]-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
methyl 3-{[(1R,3R)-3-aminocyclopentyl]sulfamoyl}thiophene-2-carboxylate
1-(2-methoxyethyl)-6-oxo-N-[(4-phenylphenyl)methyl]piperidine-3-carboxamide
6-(2-chlorophenyl)-N-(1H-imidazol-2-ylmethyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-4-[(3-fluorophenyl)methyl]piperazine
5-oxo-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
7,7-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine