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9-(2-methoxyethyl)-1-methyl-4-(pyrrolidine-1-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(1-butyl-1H-imidazol-2-yl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
{7-fluoro-5-[5-(piperidine-1-carbonyl)furan-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
3-(carbamoylmethoxy)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
4-{3-[(1E)-pent-1-en-1-yl]phenyl}-4H-1,2,4-triazole
4-({5-[1-(5-methoxypyrimidin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-chloro-3-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-9-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
ethyl 1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-5-{[({3-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)amino]methyl}-1H-pyrazole-4-carboxylate
2-[4-(2-fluorophenyl)piperazin-1-yl]-6-(2-methoxyphenyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)pyridine-3-carboxamide
N-(3-acetamido-4-methoxyphenyl)-4-(pyrrolidin-3-yl)piperazine-1-carboxamide
N-[(1R)-1-(4-methoxyphenyl)ethyl]-2-methyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
9-[(1R,2R)-2-phenylcyclopropanecarbonyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-[4-(cyclopropylmethyl)-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[(2,6-dimethoxyphenyl)methyl]-1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-amine
4-(4-methoxyphenoxymethyl)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
ethyl 1-(cyclohexylcarbamoyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-ethoxy-5-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}benzonitrile
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N,2-dimethyl-1-benzofuran-5-carboxamide
1-(2-methoxyacetyl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]piperidine-4-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetic acid
1-methyl-4-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
3-{2-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
3,3-dimethyl-1-[(3S,4R)-1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]urea
1-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-3-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}urea
1-(3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}phenyl)-1H-pyrazole
(1R,5R)-6-[(2-chloro-6-fluorophenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
1-(difluoromethyl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-1H-1,2,3-triazole-5-carboxamide
4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
2-methyl-N-[2-(4-methylmorpholin-2-yl)ethyl]-2-(thiophen-2-ylformamido)propanamide
2-[(1S,5R)-6-(2-fluoro-4-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
8-(5-chloro-2-fluorobenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-benzyl-1-(2,2-difluoroethyl)-3-ethyl-1,4-diazepan-5-one
4-methyl-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
methyl 2-[methyl({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl})amino]acetate
4-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
(1S,5R)-6-methyl-3-{[4-(methylsulfanyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-cyclopentyl-3-({1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}methyl)urea
3-{1-[(3,5-dimethyl-1H-indol-2-yl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
2-[5-(5-chlorothiophen-2-yl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-(1-methyl-1H-imidazol-2-yl)benzamide
4-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]-8-thia-4,6-diazatricyclo[7.6.0.02,7]pentadeca-1(9),2(7),5-trien-3-one
5-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
2-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
3-[1-(3-methylphenyl)piperidin-4-yl]-1-(3-sulfamoylphenyl)urea
1-ethyl-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-methylpiperidine-3-carboxamide
N4-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyrimidine-4,6-diamine
2-{[4-(methylsulfamoyl)phenyl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid