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[1-(1-ethylpiperidine-4-carbonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
2-{[3-(dimethylcarbamoyl)propyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-{1-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]ethyl}-4-methylpiperazine
4-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-({4-[6-oxo-4-(propan-2-yl)-1,6-dihydropyrimidin-2-yl]phenyl}methyl)-1λ6-thiomorpholine-1,1-dione
6-(2-chlorophenyl)-N-(3-hydroxypropyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]-1-(1-propylpiperidin-4-yl)piperidine
N-[1-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-3-phenoxypropanamide
4-(piperidin-1-ylmethyl)-N-[2-(pyridin-3-ylformamido)ethyl]benzamide
3-[(3-chlorophenyl)methyl]-1-(2,5-dimethylpyrimidin-4-yl)piperidine-3-carboxylic acid
2-(8-{[2-(furan-2-yl)phenyl]methyl}-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl)acetamide
1-cyclopentyl-4-{[2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}piperidine
1-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-1-methyl-3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}urea
4-(2-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-2-yl}ethyl)morpholine
2-(3-methoxyphenyl)-1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,5-dimethyl-1H-pyrazole-3-carboxamide
2-amino-4-(3-ethyl-1,2-oxazol-5-yl)-6-(pyridine-3-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
8-(2,5-difluorobenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-[3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-cyclohexyl-2-(methylamino)-N-(pyridin-3-ylmethyl)pyridine-4-carboxamide
(4aS,8aR)-6-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
8-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
2-[(2S)-2-amino-3-(1H-imidazol-4-yl)propanamido]-N-(pyridin-2-ylmethyl)benzamide
N-(2-methoxyethyl)-4-(1,2,3,4-tetrahydroisoquinolin-7-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3,3,3-trifluoro-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
4-(4-methoxyphenyl)-3,3-dimethyl-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperazine-1-carboxamide
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
{1-[1-(furan-3-ylmethyl)piperidin-4-yl]-2-phenylethyl}(2-methoxyethyl)(pyridin-2-ylmethyl)amine
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N,N-dimethylpyridin-2-amine
2-{5-[1-(3,5-dimethyladamantane-1-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
N-[(3-methylphenyl)methyl]-3-(2-oxooxolan-3-yl)-N-(propan-2-yl)propanamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyrimidin-2-amine
1-(1-benzothiophene-2-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
6-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonane-7-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-methyl-1-[2-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}urea
1,6-dimethyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-(methylsulfanyl)propanamide
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperidin-3-ol
7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-4-(2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-phenyl-5-(pyrazin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-fluoro-N-methyl-5-[({2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}carbamoyl)amino]benzamide
(2S,4R)-1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-4-hydroxypyrrolidine-2-carboxylic acid
(4aR,8aS)-6-(4-fluorobenzoyl)-1-[4-(morpholin-4-yl)benzoyl]-decahydro-1,6-naphthyridine
8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(3,4-dimethoxyphenyl)ethyl]-N,5-dimethyl-4-(4-methylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
5-phenyl-N-[2-(pyridin-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-methoxy-1-[1'-(5-methylthiophene-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-{[1-(pyridin-2-yl)piperidin-3-yl]methyl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
N-[2-(2-chlorophenyl)-1-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}(propan-2-yl)amine