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5-{[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]methyl}-3-phenyl-1,2,4-oxadiazole
2-[3-(5-methylfuran-2-yl)-5-[2-(morpholin-4-yl)pyrimidin-5-yl]-1H-1,2,4-triazol-1-yl]acetic acid
1-[(2,5-dimethylphenyl)methyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
6-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
4-[4-(piperidine-1-carbonyl)phenyl]phenol
8-[(2-chlorophenyl)methyl]-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
5-fluoro-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)quinazolin-4-amine
2-(2-{[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
2-(2-{[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-1-[2-(furan-2-ylmethyl)-3-hydroxypropyl]urea
6-ethyl-4-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
4-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-3-cyclopropyl-1H-1,2,4-triazol-1-yl}-3-methylpyridine
8-(4-fluoro-3-methylbenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-chloro-6-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-(tert-butylsulfamoyl)-N-[(1-methylpiperidin-3-yl)methyl]-5-{[(5-methylthiophen-2-yl)methyl]amino}benzamide
2-(4-{[ethyl(2-hydroxyethyl)amino]methyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
7-fluoro-N-(2-methoxyethyl)-3-methyl-N-[(5-methylthiophen-2-yl)methyl]-1H-indole-2-carboxamide
2-methyl-9-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
5-{[(4aS,7aR)-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-2-methyl-1H-pyrrole-3-carbonitrile
2-(2-methyl-1,3-thiazol-4-yl)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)acetamide
2-{2-[1-(1-methyl-1H-indole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
2-[4-({[3-(dimethylamino)propyl](methyl)amino}methyl)phenyl]-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
1-benzyl-N-methyl-5-({[4-(trifluoromethoxy)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-methyl-N-(2-oxopiperidin-3-yl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(2S,4R)-4-{[(3-fluorophenyl)methyl]amino}-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
2,6-dimethoxy-3-[2-(pyridin-2-yl)piperidine-1-carbonyl]pyridine
3-(2,4-dimethoxybenzoyl)-1-[(2,5-dimethoxyphenyl)methyl]piperidine
{4-[4-(1H-imidazol-1-ylmethyl)phenyl]phenyl}methanol
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(1H-indol-3-yl)ethan-1-one
3-[(3R,4S)-1-(4-methoxy-2-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
5-{2-oxo-2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-(azepan-1-yl)-3-[4-chloro-2-({[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
9-hydroxy-3-[2-(3-methoxypropyl)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
3-(azocan-1-yl)-1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]propan-1-one
3-{5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
(2-{2-[1-(3,4-difluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
4-(4-propyl-1,4-diazepan-1-yl)-N-(pyridin-4-ylmethyl)pyridine-2-carboxamide
5-{imidazo[1,2-a]pyridine-6-carbonyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-methyl-2-[4-(morpholin-4-yl)-2-{[2-(1,3-thiazol-4-yl)ethyl]amino}pyrimidin-5-yl]propanoic acid
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
N3-{[1-(2-fluorophenyl)cyclopentyl]methyl}piperidine-1,3-dicarboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-(thiophen-2-ylmethyl)piperidine-3-carboxamide
5-tert-butyl-N-[(5-methylpyrazin-2-yl)methyl]-1,3,4-oxadiazol-2-amine
3-(pentan-2-yl)-8-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2-methoxyacetyl)-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]piperidine-4-carboxamide
4-[2-(3-fluorophenyl)ethyl]-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(3S,5S)-1-(3-phenylpropyl)-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid