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4-(3-cyclohexylpyrrolidine-1-carbonyl)-1-(diphenylmethyl)-1H-1,2,3-triazole
1-(3,5-dimethylphenyl)-4-(3-ethoxypropanoyl)piperazin-2-one
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-cyclohexylpiperazin-2-yl]ethan-1-ol
4-(hydroxymethyl)-1-(1-methyl-1H-indole-3-carbonyl)azepan-4-ol
2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-7-methyl-1H-1,3-benzodiazole
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(2-oxopyrrolidin-1-yl)acetamide
1-(4-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}thiophen-2-yl)ethan-1-one
methyl (2S)-2-[(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}phenyl)formamido]-3-methylbutanoate
1-[3-(1H-imidazol-1-yl)propyl]-5-[(E)-2-(2-methoxyphenyl)ethenyl]-4-phenyl-1H-imidazole
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-(pyrrolidin-3-yl)ethan-1-one
ethyl 1-(4-methyl-1,3-thiazole-5-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
3-(pyrrolidin-1-yl)-1-(thiophen-3-ylmethyl)piperidine
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
2-{[7-(4-methylpentanoyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}benzonitrile
(3S,5R)-1-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-5-(cyclopropylcarbamoyl)piperidine-3-carboxylic acid
4-[(2-chloro-4-fluorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
5-{1-[2-(2-fluoro-4-methoxyphenyl)-1H-imidazol-1-yl]-2-methylpropyl}-1-methyl-1H-1,2,4-triazole
1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-6-oxo-N-propylpiperidine-3-carboxamide
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{1-oxaspiro[4.5]decan-3-yl}propanamide
5-ethyl-N4-[2-(piperidin-1-yl)ethyl]pyrimidine-2,4-diamine
3-(2,6-dimethylphenoxy)-N-(1-methyl-1H-1,2,3-benzotriazol-5-yl)azetidine-1-carboxamide
1-(pyridin-4-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepane
3-methyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}furan-2-carboxamide
7-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]-1,2-dihydroisoquinolin-1-one
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
(3S,4R)-1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
3-chloro-N-({1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)thiophene-2-carboxamide
N-cyclopropyl-1-{1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]piperidin-4-yl}piperidine-3-carboxamide
ethyl 4-benzyl-1-(1H-indol-2-ylmethyl)piperidine-4-carboxylate
4-{4-[1-(oxolan-2-ylmethyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine
1-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-(morpholin-3-yl)ethan-1-one
(3S,4R)-1-(1-carbamoylcyclopropanecarbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,4,5-trifluorobenzamide
N4-[(3-fluorophenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
2-{[4-(2,6-dimethylphenyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
dimethyl({4-methyl-5-[1-(2-methylquinolin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
2-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-4,6-dimethylpyridine-3-carbonitrile
N-butyl-N-[(5-methylthiophen-2-yl)methyl]oxane-2-carboxamide
7-[2-(pyridin-3-yl)quinoline-4-carbonyl]-2-oxa-7-azaspiro[4.5]decane
N-[2-(azepan-1-yl)-2-phenylethyl]-1-cyclopropyl-1H-pyrrole-2-carboxamide
1-{4-[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]piperidin-1-yl}ethan-1-one
[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl][1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxy-2-methylpropan-1-one
2-(adamantan-1-yl)-N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}acetamide
N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}isoquinoline-3-carboxamide
3-[2-(3-fluorophenyl)ethyl]-1-(furan-3-carbonyl)piperidine
4-[(2-ethoxyphenyl)methyl]-3-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-2-one
N-[(3R,4R)-1-(1,3-benzoxazol-2-yl)-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
1-(3-carbamoylpyridin-2-yl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine