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1-(2,3-dihydro-1H-inden-2-yl)-N-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}piperidin-3-amine
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
6-(2,5-dimethylfuran-3-yl)-2-[(3S)-3-hydroxypyrrolidine-1-carbonyl]-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(4-methylphenoxy)ethan-1-one
4-{5-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(pyrimidin-4-ylmethyl)acetamide
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-[(4-hydroxyazepan-4-yl)methyl]-2-phenylbenzamide
(4aR,8aS)-1-[(4-fluorophenyl)methyl]-6-(furan-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
4-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)piperazine-2-carboxylic acid
N-phenyl-5-[3-(pyridin-3-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(1-{5-methyl-4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]thieno[2,3-d]pyrimidine-6-carbonyl}piperidin-4-yl)methanol
4-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
3-({2-methyl-3-[(pyridin-2-ylmethyl)amino]phenyl}formamido)-N-(2-methylphenyl)propanamide
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(3-methylpyridin-4-yl)-1,4-diazepane
2-{3-[(4-hydroxypiperidin-1-yl)methyl]phenyl}-6-(2-methyl-1,3-thiazol-4-yl)-3,4-dihydropyrimidin-4-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]benzamide
1-ethyl-N-[2-(4-methoxyphenyl)ethyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2R,3R)-3-amino-1'-[2-(dimethylamino)benzoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-[(3-methylphenyl)sulfanyl]-1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperidine
8-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole-5-carbonyl]-1-oxa-8-azaspiro[4.5]decane
2-ethoxy-N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]pyridine-3-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
(4aS,8aR)-6-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
2-(1H-indazol-3-yl)-1-(1,2-oxazinan-2-yl)ethan-1-one
6-methyl-5-(2,3,4-trimethoxyphenyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2S,4R)-4-(2-cyclopentylacetamido)-N-ethyl-1-[(3-hydroxyphenyl)methyl]pyrrolidine-2-carboxamide
N4-ethyl-N4-methyl-N2-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrimidine-2,4-diamine
8-[3-(5-methylfuran-2-yl)butyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methyl-7-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
N-(butan-2-yl)-5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
N-(cyclopropylmethyl)-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
4-methyl-2-[1-(pyridine-3-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
2-[3-(1-benzofuran-2-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
4-({5-[4-(methoxymethyl)-5-methyl-1,2-oxazol-3-yl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
4-hydroxy-N-(2-methoxyethyl)-2-(pyridin-2-yl)-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
N-(2-chlorophenyl)-3-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}propanamide
3-{[4-(2-methylphenyl)-1,4-diazepan-1-yl]methyl}piperidin-3-ol
{1-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl}methanamine
1-[2-(cyclohex-1-en-1-yl)ethyl]-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
6-ethyl-2-methyl-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]quinoline-4-carboxamide
1-(3-fluoropyridin-4-yl)-4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazine
1-[1-(1H-indole-6-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
1-(2,1,3-benzothiadiazol-4-yl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methylurea
2-(1-benzylpiperidin-4-yl)-1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]ethan-1-one
(1S,6R)-9-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
[(3R,4R)-1-(6-cyclopropylpyrimidin-4-yl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N2,N4-dimethylpyrimidine-2,4-diamine