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2-{[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]amino}-N-[(2-fluorophenyl)methyl]acetamide
2-{3-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]piperidin-1-yl}acetamide
2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]-1-[4-(pyridin-3-yl)piperazin-1-yl]ethan-1-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(2-methoxyphenyl)acetamide
N-[(4-methoxyphenyl)methyl]-4-methyl-2-oxo-N-propylpentanamide
N-{2-[4-(furan-2-ylmethyl)morpholin-2-yl]ethyl}-1,3-thiazole-5-carboxamide
4-[(2-fluoro-4-methoxyphenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}pyridine
1-(5-chloropyridin-2-yl)-4-(2,3-dihydro-1-benzofuran-5-carbonyl)piperazine
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-ethoxyethan-1-one
6-methoxy-N-methyl-2-oxo-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
6-{1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-carbonyl}-2,3,4,9-tetrahydro-1H-carbazole
(2S,4S)-4-amino-1-[2-(2,3-dihydro-1H-indol-1-yl)-2-oxoacetyl]-N,N-diethylpyrrolidine-2-carboxamide
1-(3-chlorophenyl)-4-(thiophene-3-carbonyl)piperazin-2-one
(2S)-2-hydroxy-4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]formamido}butanoic acid
1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(pyridin-2-yl)piperidin-4-ol
4-[1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)azetidin-3-yl]pyridine
5-cyclopropyl-N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-1,3,4-oxadiazol-2-amine
1-[(4-chlorophenyl)methyl]piperidin-3-amine
(4aS,7aR)-1-[4-(1H-imidazol-1-yl)butanoyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(3,4-dimethoxyphenyl)-5-[4-hydroxy-1-(pyridin-3-ylmethyl)piperidin-4-yl]-1-benzofuran-2-carboxamide
1-(2-methoxy-5-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
1-{2-methoxy-5-[(4-methylpiperidin-1-yl)methyl]phenoxy}-3-(piperidin-1-yl)propan-2-ol
5-{[4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]methyl}-3-(propan-2-yl)-1,2-oxazole
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2-methoxybenzamide
2-(3,3,3-trifluoropropanoyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
5-(2-{4-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-1H-1,2,3-triazol-1-yl}ethyl)-1,3,4-thiadiazol-2-amine
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-{[(4,8-dimethoxynaphthalen-1-yl)methyl](methyl)amino}propane-1,2-diol
methyl 4-{5-amino-4-cyano-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-trien-3-yl}thiophene-2-carboxylate
(2S)-3-(1H-imidazol-4-yl)-2-[4-phenyl-5-(propan-2-yl)-1H-imidazol-1-yl]propanoic acid
3-{[2-(5-propylfuran-2-yl)-1H-imidazol-1-yl]methyl}pyridine
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
4-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-1λ6-thiomorpholine-1,1-dione
3-phenyl-3-(pyridin-2-yl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}propanamide
1-(4-aminopyrimidin-2-yl)-4-(1,3-thiazol-2-ylmethyl)-1,4-diazepan-6-ol
4-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
4-hydroxy-2-methyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]pyrimidine-5-carboxamide
1-(6-hydroxy-4-{[3-(4-methoxyphenoxy)phenyl]methyl}-1,4-diazepan-1-yl)ethan-1-one
N,1-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1H-indole-3-carboxamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(5-methylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-{1-[(2-ethoxyphenyl)methyl]-4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
3-methyl-4-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethoxy]-1,2,5-oxadiazole
2-hydroxy-5-({2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)benzoic acid
{4-[(2-chlorophenyl)methyl]-1-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl}methanol
(3R,4R)-1-[(2-chloro-4-fluorophenyl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
2-butyl-N-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-2,5-dihydro-1H-pyrrole-1-carboxamide
N,N-dimethyl-3-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]aniline