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1-[(3S)-3-ethylmorpholin-4-yl]-2-[(3-methoxyphenyl)sulfanyl]ethan-1-one
3-(5-{2-[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-1,2,4-triazol-3-yl)pyridine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-1H-1,2,3-benzotriazole-5-carboxamide
1-cyclopentyl-4-[2-(2,4-dichlorophenoxy)acetyl]piperazin-2-one
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]pyrrolidin-3-yl]urea
(3S)-2-[(2-aminopyridin-3-yl)methyl]-N-tert-butyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-benzyl-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]piperazine-1-carboxamide
(2R,6S)-4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,6-dimethylmorpholine
2-[1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)piperidin-3-yl]-1,3-benzoxazole
{4-[3-(trifluoromethyl)pyridin-2-yl]-1,4-oxazepan-6-yl}methanol
N-(1-benzothiophen-2-ylmethyl)-N-methyl-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]thiomorpholine
1-{1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}-N,N-dimethylpyrrolidin-3-amine
5-methyl-3-[(6-methylpyridin-2-yl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
methyl 2-hydroxy-5-({4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-1-yl}methyl)benzoate
2-methyl-6-{1-[4-(pyridin-2-yl)pyrimidin-2-yl]piperidin-4-yl}pyrimidin-4-ol
2-[2-benzyl-5-oxo-4-(2-phenylphenyl)piperazin-1-yl]acetamide
1-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
6-{[4-(1-methylpiperidin-4-yl)piperazin-1-yl]methyl}naphthalen-2-ol
4-(3-phenoxybenzenesulfonyl)piperazine-2-carboxylic acid
1-{4-[3-({[(3-chloro-4-ethoxyphenyl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
3-(2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindol-1-one
N-ethyl-4-methyl-5-[3-(oxan-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-1,3-thiazol-2-amine
{3-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]-3-phenylpropyl}dimethylamine
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
N-ethyl-6-[4-(hydroxymethyl)phenyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
N-[(3-methyl-1-benzofuran-2-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-3-(2-oxopiperidin-1-yl)propanamide
8-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-2,8-diazaspiro[4.5]decan-3-one
1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-4-(4-methylphenoxy)piperidine-4-carboxylic acid
2-(4-phenylmethanesulfonylmorpholin-3-yl)-1-(thiomorpholin-4-yl)ethan-1-one
2-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)benzoic acid
3-{2-[2-(1-benzothiophen-2-yl)-1H-imidazol-1-yl]ethyl}-4-methyl-4H-1,2,4-triazole
3,5-dichloro-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-(prop-2-en-1-yloxy)benzamide
4,5-dimethyl-6-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrimidin-2-amine
3-{[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]methyl}-4H-chromen-4-one
1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
4-methyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-1,2,5-oxadiazole-3-carboxamide
3-(2-fluoro-3-methoxyphenyl)-5,6-dimethyl-1,2-dihydropyridin-2-one
6-(2,5-dimethylfuran-3-yl)-N-(1-methyl-2-oxopyrrolidin-3-yl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-[1-(oxane-4-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
N-methyl-N'-(2-methylphenyl)-N-[2-(2-oxopiperidin-1-yl)ethyl]propanediamide
N-cyclohexyl-2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-cyclopropyl-2-[4-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)piperidin-1-yl]acetamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-{3-[(3-fluorophenyl)methoxy]benzoyl}pyrrolidin-3-yl]methanol
tert-butyl(furan-2-ylmethyl){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
8-{2-[(2-methylphenyl)sulfanyl]acetyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}cyclohexanecarboxamide