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3-[4-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazol-1-yl]propane-1,2-diol
1-[2-(3-methoxyphenyl)azetidin-1-yl]-2-(1-methylpiperidin-4-yl)ethan-1-one
N-(5-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-2-methylphenyl)cyclopropanecarboxamide
(1R,9aR)-1-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
2-(methylamino)-N-[3-(4-methylpiperidin-1-yl)-3-oxopropyl]pyridine-3-carboxamide
2,6-difluoro-N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}benzene-1-sulfonamide
1-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine
6-cyclopentyl-N,1-dimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-phenylpiperidine-4-carbonitrile
(1-{1-[1-(2-phenylethyl)piperidin-4-yl]piperidin-3-yl}piperidin-4-yl)methanol
5-(2-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-methyl-5-{1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1,2-oxazole
4-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2,6-dimethoxyphenol
1-(2-{[4-(2-methoxyethoxy)piperidin-1-yl]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
7-fluoro-2-methyl-4-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]quinoline
N-[(3-hydroxypiperidin-3-yl)methyl]-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]pyrimidin-2-amine
1-(cyclohexylmethyl)-4-oxo-N3-(propan-2-yl)-N5-[2-(pyridin-4-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(pyridin-2-ylmethyl)acetamide
2-methyl-5-(propan-2-yl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-ethyl-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxamide
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-5-(4-fluorophenyl)-1,2,4-triazin-3-amine
(2R)-2-(cycloheptylamino)-3-phenylpropan-1-ol
8-methoxy-N-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
1-(4-{2-[4-(3-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
8-[(3-hydroxyphenyl)methyl]-3-(2-methoxyethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R)-1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-(pyridine-3-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
6-methoxy-3-methyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1-benzofuran-2-carboxamide
5-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
2-ethoxy-5-{1-[(1-methylpiperidin-2-yl)methyl]-1H-imidazol-2-yl}pyridine
(4aR,8aS)-6-cyclohexyl-1-(cyclohexylmethyl)-decahydro-1,6-naphthyridin-2-one
4-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}pyridine
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-(2,5-dimethylphenyl)-N'-methyl-N'-(oxan-2-ylmethyl)propanediamide
[(3R,4R)-1-(6-ethyl-2-methylpyrimidin-4-yl)-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-[2-(pyrrolidin-1-yl)ethyl]urea
2,4-dimethoxy-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}benzene-1-sulfonamide
2-chloro-N-{2-[3-(morpholin-4-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}benzamide
1-[(4-methoxypyridin-2-yl)methyl]-1,2-dihydroquinolin-2-one
2-(4-{[4-(difluoromethoxy)phenyl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
9-[(3-ethenylphenyl)methyl]-3,9-diazaspiro[5.6]dodecane
(3aS,6aS)-5-[(6-methoxynaphthalen-2-yl)methyl]-octahydropyrrolo[3,4-b]pyrrole
3-{[(2-{[3-(trifluoromethyl)phenyl]methoxy}-6H,7H,8H-cyclopenta[g]quinolin-3-yl)methyl]amino}-1λ6-thiolane-1,1-dione
1-(diphenylmethyl)-4-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
2-(2-aminoethyl)-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}quinazolin-4-amine
1-[7-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-4-ol
N-(2-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-yl}-2-oxoethyl)methanesulfonamide
N-benzyl-N-(cyclobutylmethyl)-2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3,5-dimethyl-2-({[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)pyridin-4-ol