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2-chloro-N-(2-{[5-oxo-1-(propan-2-yl)pyrrolidin-3-yl]formamido}ethyl)benzamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
(1S,5R)-3-[(6-chloro-2H-chromen-3-yl)methyl]-3,9-diazabicyclo[3.3.2]decan-10-one
4-({3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}methyl)-2,1,3-benzothiadiazole
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amine
3-amino-1-{[2,5-dimethyl-1-(4-methylpyridin-2-yl)-1H-pyrrol-3-yl]methyl}pyrrolidine-3-carboxylic acid
1-({3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,4-dihydroquinolin-4-one
2-{[4-(carboxymethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-methyl-6-[2-(morpholin-4-yl)ethyl]-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
1-cyclopropyl-6-oxo-N-[(1-phenylcyclopentyl)methyl]piperidine-3-carboxamide
N-(4-cyanophenyl)-4-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]butanamide
2-(3-methylphenoxy)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethan-1-one
8-cyclopropanecarbonyl-2-[(5-methylthiophen-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(2H-1,2,3-benzotriazol-2-yl)-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
(2S,4R)-4-amino-1-{3-[(3-ethylphenyl)carbamoyl]propanoyl}-N-methylpyrrolidine-2-carboxamide
7-fluoro-3-{[(6-methyl-2-propylpyrimidin-4-yl)amino]methyl}-1,2-dihydroquinolin-2-one
N-(1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-4-carboxamide
1-(3-chloro-4-methoxyphenyl)-3-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]urea
4-(2,3-dihydro-1H-inden-5-yloxy)-1-(5-fluoropyridin-2-yl)piperidine-4-carboxylic acid
2-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}thiophene-3-sulfonamide
2-(3-methylbutyl)-8-(1H-pyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-2-amine
2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1,3-oxazole
5-[1-(2-methyl-1,3-benzothiazol-6-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(1-oxo-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-2-yl)pyrrolidin-2-one
3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1-[3-(2-methoxyphenyl)phenyl]urea
N-(2-fluoroethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
1-[(5-methylfuran-2-yl)methyl]-4-oxo-N3-(prop-2-en-1-yl)-N5-{[3-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
(3R,4R)-4-(morpholin-4-yl)-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-3-ol
(4S)-1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-3,3,4-trimethylpiperidin-4-ol
2-methyl-N-(2-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyridin-3-yl)propanamide
2-{2-[1-(quinoline-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
4-ethyl-1-methyl-3-(1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aS,6aS)-2-methyl-5-[(2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)sulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-hydroxy-2-phenylpyrimidine-5-carbonyl)piperidine-3-carbonitrile
3-methyl-2-(3-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyridine
1-[2-(dimethylamino)-2-(3-fluorophenyl)acetamido]cyclopentane-1-carboxamide
2-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
3-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pent-2-yn-1-yl)pyrrolidin-3-yl]-1H-pyrazole-5-carboxamide
1-methyl-8-[2-(2-oxopyrrolidin-1-yl)ethyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-N-[(3R)-pyrrolidin-3-yl]acetamide
1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
1-[1-(2H-1,3-benzodioxol-5-yl)-3-(propan-2-yl)-1H-1,2,4-triazole-5-carbonyl]-2-methylpiperidine
(benzylsulfamoyl)[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]amine
1-ethyl-N-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]thiomorpholine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methyloxane-2-carboxamide