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ethyl 1-[2-(pyridin-3-yl)ethyl]-1H-imidazole-2-carboxylate
3-[4-(1H-pyrazol-1-yl)phenyl]-5-(pyrrolidine-1-sulfonyl)benzoic acid
N-cyclopropyl-3-{1-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
N4-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
1-ethyl-5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-3-(2-methylpropyl)-1H-pyrazole
N4-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(2S,4R)-1-benzyl-N-methyl-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
benzyl({[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl})(cyclopropylmethyl)amine
1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-[(2-methylphenyl)sulfanyl]piperidine
1,4-dimethyl-N-[2-(3-propoxyphenyl)ethyl]piperidine-4-carboxamide
(2S,4R)-N-ethyl-4-{4-[({[(3-methylphenyl)methyl]carbamoyl}amino)methyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxamide
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]propanamide
5-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-benzotriazole
4-ethyl-N,N-dimethyl-6-(1H-pyrazol-4-yl)pyrimidin-2-amine
N-[2-(3-chlorophenyl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-({2-[(3-methoxyphenyl)methyl]morpholin-4-yl}methyl)-1H-1,3-benzodiazole
2-[4-(1H-indol-2-ylmethyl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
2-(2,4-dimethoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-({4-[(3S)-3-fluoropyrrolidine-1-carbonyl]phenyl}methyl)-3,5-dimethyl-1H-pyrazole
5-(3-methoxyphenoxymethyl)-3-(2-phenylazetidine-1-carbonyl)-1H-pyrazole
(1R,2R)-2-{4-[1-(2-phenylethyl)-1,2,3,6-tetrahydropyridin-4-yl]-1H-pyrazol-1-yl}cyclohexan-1-ol
N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}furan-2-carboxamide
N-methyl-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-(quinolin-5-ylmethyl)propanamide
8-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
ethyl 4-{1-[(6-chloroquinolin-2-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
2-[2-(2,4-dimethylphenoxy)ethyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
N-[4-(6-chloropyridin-3-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]-2-(dimethylamino)acetamide
propyl 2-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]acetate
2-amino-N-[(3,5-difluoro-4-methoxyphenyl)methyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
8-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]acetamide
4-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-N,N-dimethyl-4-oxobutanamide
5-ethyl-7-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}pyrazolo[1,5-a]pyrimidine
2-{benzyl[1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}ethan-1-ol
5-amino-N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
5-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-2-methylphenol
{2-[2-(1-cyclopentanecarbonylpiperidin-3-yl)-1H-imidazol-1-yl]ethyl}dimethylamine
(3S)-1-[(5-cyclohexylthiophen-2-yl)methyl]pyrrolidin-3-amine
1-[1-(7-fluoroquinazolin-2-yl)piperidin-4-yl]-1,4-diazepan-6-ol
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-2-methyl-2-(morpholin-4-yl)propan-1-one
2-cyclopropyl-6-{[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyrimidin-4-ol
1-{[5-(cyclohex-3-en-1-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-4,4-difluoropiperidine
3-(dimethyl-1,2-oxazol-4-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-1-one
(1S,5R)-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
9-[3-(4-hydroxyphenyl)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
(3S,7S)-5-(2-fluorobenzoyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
3-[2-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-4-[(2-ethoxyphenyl)methyl]piperazin-2-one
[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl][(4-methoxy-2,3-dimethylphenyl)methyl]methylamine
N-methyl-3-propyl-N-(quinoxalin-2-ylmethyl)-1H-pyrazole-5-carboxamide
1-({5-[1-(4-hydroxybutyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol