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1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(2-methoxybenzoyl)piperazine
N-methyl-4-oxo-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1'-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N,N-dimethyl-1-[4-(4-methylphenyl)-5-(pyrimidin-5-yl)pyrimidin-2-yl]pyrrolidin-3-amine
5-chloro-N-{2-[1-(propan-2-yl)piperidin-3-yl]ethyl}thiophene-2-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(2-methoxyphenyl)-N-[1-(pyridin-2-yl)propan-2-yl]benzamide
1-[benzyl(methyl)amino]-3-(2-methoxy-5-{[(1-phenylcyclopropyl)amino]methyl}phenoxy)propan-2-ol
5-(2,2-diethylmorpholine-4-carbonyl)-1-(pyridin-2-ylmethyl)piperidin-2-one
4-[(3-fluorophenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-2-(methylamino)acetamide
2-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenoxy)pyrimidine
3-hydroxy-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyridine-2-carboxamide
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
4-[(2-methyl-1H-imidazol-1-yl)methyl]-1-(1-methyl-1H-imidazole-2-carbonyl)piperidine
4-(hydroxymethyl)-1-(1-phenylcyclohexanecarbonyl)azepan-4-ol
5-(methoxymethyl)-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)thiophene-2-carboxamide
6-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-4-yl)-2-methylpyrimidin-4-ol
3-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
(2-{[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](thiophen-3-ylmethyl)amino}ethyl)dimethylamine
{3-[2-({dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)ethyl]-1,2,4-oxadiazol-5-yl}methanol
(1S,5R)-6-[3-(1H-imidazol-2-yl)benzoyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-methyl-4-[5-(4-methyl-1,2,5-oxadiazol-3-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]pyridine
2-cyclopropyl-8-[(2,5-dimethylthiophen-3-yl)sulfonyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(oxolan-2-ylmethyl)-2-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenoxy)acetamide
(2S,3R)-2-amino-1-[3-(3-ethylphenoxy)azetidin-1-yl]-3-hydroxybutan-1-one
5-[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
(1S,5R)-3-cyclobutanecarbonyl-6-(1-methyl-1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2,6-dimethyl-3-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,4-dihydropyridin-4-one
N-[(1-ethylcyclobutyl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
3-(azepane-1-carbonyl)-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(4-{3-[(4-hydroxyphenyl)methyl]-4H-1,2,4-triazol-4-yl}phenyl)ethan-1-one
3-(3-hydroxy-3-methylbutyl)-N-(pyridin-3-ylmethyl)benzamide
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
6,7-dimethoxy-3-[(2,4,5-trifluorophenyl)methyl]-3,4-dihydroquinazolin-4-one
methyl 9-[2-(2-fluorophenyl)ethoxy]-7-oxo-3-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N5-cyclopropyl-N6-[2-(methylsulfanyl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
(4aS,8aR)-1-(2-aminoethyl)-6-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-decahydro-1,6-naphthyridin-2-one
(4aS,7aR)-1-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(2,4-dimethoxypyrimidin-5-yl)isoquinoline
7-(3-chlorophenyl)-4-[(3-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-9H-purin-6-amine
N-[(4-fluorophenyl)methyl]-3-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]propanamide
(3R)-N-(4-chloro-2-ethylphenyl)-3-hydroxypyrrolidine-1-carboxamide
5-(oxolan-2-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}thiophene-2-carboxamide
3-(3-fluorophenyl)-4-[1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]piperazin-2-one
4-{4-[2-(2-methylphenyl)acetyl]piperazin-1-yl}-2-(naphthalen-1-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-amino-N-cyclohexyl-N-methyl-1,3-benzothiazole-5-carboxamide