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1-{5-[2-(dimethylamino)phenyl]-1H-1,3-benzodiazol-2-yl}ethan-1-ol
3-ethyl-N-[3-(2-methoxyphenyl)propyl]-1H-pyrazole-4-carboxamide
(4S)-1-(6-aminopyridine-3-carbonyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
2-[3-(1H-imidazol-1-yl)propyl]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1-oxo-2,3-dihydro-1H-isoindole-5-carboxamide
N-[2-(ethylsulfanyl)ethyl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-ethyl-1-methyl-5-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrazole
(3S,9aR)-3-(hydroxymethyl)-2-methyl-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-methanesulfonyl-2,7-diazaspiro[4.5]decane
2-amino-4-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]-6-(3,4,5-trifluorophenyl)pyridine-3-carbonitrile
N-[3-({ethyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]carbamoyl}amino)-4-methoxyphenyl]acetamide
(4aS,8aR)-1-(4-hydroxybutyl)-6-(4-methyl-1H-imidazole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
ethyl 4-(1-methyl-4-oxo-1,4-dihydroquinoline-3-amido)piperidine-1-carboxylate
1-(6-methyl-2-propylpyrimidin-4-yl)-N-(pyridin-2-ylmethyl)piperidin-4-amine
methyl (2S,4S,5R)-5-(3-chlorophenyl)-4-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}-1-methylpyrrolidine-2-carboxylate
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,N-dimethyl-4-oxobutanamide
ethyl 4-(1-cycloheptyl-6-oxopiperidine-3-amido)piperidine-1-carboxylate
1-{[4-(pyridin-4-yl)thiophen-2-yl]methyl}piperazine
4-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(4-ethoxyphenyl)methyl]-N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}cyclopropanamine
7-(3-methoxyphenyl)-2-(5-methyl-1H-1,2,4-triazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[1-(2,5-dimethylphenyl)-5-(6-oxopiperidin-3-yl)-1H-1,2,4-triazol-3-yl]acetamide
methyl 3-(2-chloro-6-fluorobenzamido)-6-[(4-methylpiperidin-1-yl)methyl]thieno[2,3-b]pyridine-2-carboxylate
4-(4-fluorophenyl)-1-[2-(pyrrolidin-1-yl)pyrimidine-5-carbonyl]piperidin-4-ol
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
4-[(3,3-dioxo-1,3λ6,4-oxathiazinan-4-yl)methyl]-N-methylbenzamide
1-{4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}-2-(2-methylphenyl)ethan-1-one
2-cyclopropyl-9-(6-methyl-2-propylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
1-[2-(3-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
1-(furan-3-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
4-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}morpholine
(3S,4S)-1-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-ethyl-8-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(2S,4R)-4-(dimethylamino)-1-(2-ethylbenzoyl)pyrrolidine-2-carboxylic acid
7-[2-chloro-4-(1H-pyrazol-1-yl)benzoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
6-methyl-2-{1-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
4-(pyridin-3-yl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}pyrimidin-2-amine
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
1-{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}piperidin-3-ol
N-(2H-1,3-benzodioxol-5-yl)-1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperidin-3-amine
(3R,5S)-1-benzyl-N-[2-(1H-imidazol-4-yl)ethyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}piperidine-3-carboxamide
8-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3-chlorophenyl)methyl]-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
ethyl 5-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(2-methyl-3-{methyl[1-(1,3-thiazol-2-yl)ethyl]carbamoyl}phenyl)oxolane-2-carboxamide
5-butyl-1-(2-methoxyphenyl)-4-(pyridazine-3-carbonyl)piperazin-2-one
N-(2-ethoxyphenyl)-N'-[4-(pyridin-2-yl)butyl]propanediamide
2-({4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}sulfanyl)ethan-1-ol
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-[1-(1H-pyrazol-3-ylmethyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine