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N-(4-acetylphenyl)-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
methyl 5-[(4-hydroxy-4-methylpentan-2-yl)amino]-3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[(2R)-2-aminopropanoyl]-N-[4-(1,3-benzoxazol-2-yl)phenyl]piperidine-4-carboxamide
1-[2-(5-{imidazo[2,1-b][1,3]thiazol-6-yl}-1,2,4-oxadiazol-3-yl)ethyl]-4-methylpiperazine
N-[(3-ethoxy-4-methoxyphenyl)methyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(furan-2-ylmethyl)-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]piperidine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
3-[4-(2-chlorophenoxy)piperidine-1-carbonyl]-5-fluorobenzonitrile
3-(2-amino-1,3-thiazol-4-yl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
N-[1-(4-fluorophenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]oxolane-3-carboxamide
5-(1H-imidazol-1-ylmethyl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}furan-2-carboxamide
methyl N-{2-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}carbamate
ethyl 4-(2-phenylethyl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine-4-carboxylate
1'-(8-hydroxyquinoline-7-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2,2-dimethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}propanamide
1-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-benzyl-4-(4-methylpyridin-2-yl)-1,4-diazepan-6-ol
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
2-[2-methyl-3-(1H-1,2,4-triazol-1-yl)propanamido]-N-[2-(morpholin-4-yl)ethyl]benzamide
7-(pyridin-2-ylmethyl)-4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
(4aS,8aR)-1-(3-hydroxypropyl)-6-(3,3,3-trifluoropropyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)acetamide
1-[4-(4-fluorophenoxy)piperidin-1-yl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
7-methoxy-N-{3-[(pyridin-3-yl)amino]propyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
7-(cyclopropylmethyl)-2-{[2-(trifluoromethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
N-ethyl-2-[4-(5-phenyl-1,2,4-oxadiazol-3-yl)piperazin-1-yl]acetamide
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-methylpropanamide
3-benzyl-4-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]piperazin-2-one
6-tert-butyl-1-methyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[3-(oxan-4-yl)-5-[(oxolan-2-ylmethoxy)methyl]-1H-1,2,4-triazol-1-yl]pyridine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2-hydroxy-2-phenylethyl)-N-methylbenzamide
(1R,7S)-3-[2-(pyridin-4-yl)ethyl]-6-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-(4-fluorophenyl)-1-(quinoline-6-carbonyl)piperidin-3-amine
(1S,5R)-3-(4-methylpiperazine-1-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(pyridin-2-yl)propan-1-one
5-{3-[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]propyl}-1H-1,2,3,4-tetrazole
(7R,9aR)-N-cyclohexyl-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
3-benzyl-4-(2-methoxy-5-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aR,6aR)-2-cyclopropanecarbonyl-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-cyclopentyl-N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methylpyrimidin-2-amine
4-[4-(benzenesulfonyl)piperazin-1-yl]-5,6,7,8-tetrahydroquinazolin-2-amine
2-(4-fluoro-3-methoxyphenyl)-1-[1-(4-methanesulfonylphenyl)ethyl]-1H-imidazole
(2S)-4-(methylsulfanyl)-2-{[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}butan-1-ol
1-{2-methyl-5-[2-(pyridin-2-yl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
3-{2-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]ethyl}-1,3-oxazinan-2-one
N-(3-fluoro-2-methylphenyl)-2-{[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]amino}acetamide
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-4-methoxycyclohexane-1-carboxamide