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N-benzyl-2,5-dimethyl-N-(1,3-thiazol-2-ylmethyl)-1,3-thiazole-4-carboxamide
1-ethyl-4-{[3-(3-methoxypropyl)piperidin-1-yl]methyl}-1H-indole
ethyl 3-{3-[(2-fluorophenyl)formamido]propanamido}-4-methylpentanoate
5-ethanesulfonamido-N,1-dimethyl-2-phenyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
6-ethyl-N,1-dimethyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
[(2S,6S)-11-methoxy-4-(2-methyl-5-propylpyrimidin-4-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
3-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidine-1-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
5-methyl-1-(2-methylphenyl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperazin-2-one
(3aS,6aS)-N-(5-fluoro-2-methylphenyl)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carboxamide
6-(piperidin-1-yl)-N-[2-(1H-1,2,3-triazol-1-yl)ethyl]pyrimidin-4-amine
methyl 1-[1-benzyl-2-methyl-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carbonyl]piperidine-4-carboxylate
N-butyl-N-(3-phenylprop-2-yn-1-yl)-6-azaspiro[2.5]octane-1-carboxamide
5-methyl-4-[(2-methyl-1H-imidazol-1-yl)methyl]-2-(naphthalen-2-yl)-1,3-oxazole
N-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]-2-(2-methyl-1H-imidazol-1-yl)acetamide
2-(1H-indazol-3-yl)-N-{1-oxaspiro[4.4]nonan-3-yl}acetamide
4-[(3-fluorophenyl)methyl]-1-(1-phenylcyclopropanecarbonyl)-1,4-diazepan-5-one
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-(piperidin-1-yl)piperidine-4-carboxamide
methyl 6-[2-({2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamido}methyl)-2,3-dihydro-1-benzofuran-7-yl]pyridine-3-carboxylate
(1R,9aR)-1-[2-(1,2-oxazol-5-yl)phenoxymethyl]-octahydro-1H-quinolizine
1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(3-methylthiophen-2-yl)-1H-imidazole
1-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]-1-methylurea
5-(2,6-difluorophenyl)-3-(ethoxymethyl)-1-ethyl-1H-1,2,4-triazole
(3S,4S)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
2-[(3R)-3-hydroxypyrrolidine-1-carbonyl]-6-(4-methoxyphenyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
5-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N,N-dimethylpyridin-2-amine
(2S)-2-amino-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
1-{3-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
2-(2,3-dimethylphenoxy)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
6-[3-(3-hydroxy-3-methylbutyl)benzoyl]-2-methyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-(2-hydroxybutyl)-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
7-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]-3-methyl-3,4-dihydroquinazolin-4-one
3-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-(5-methylpyridin-3-yl)urea
1-(3-methylfuran-2-carbonyl)-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
3,3-dimethyl-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
4-[4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]-1-[(4-methylphenyl)methyl]pyrrolidin-2-one
2-(2-chloro-4-{[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]methyl}-6-methoxyphenoxy)acetic acid
8-[(3,4,5-trifluorophenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylacetamide
3-{3-[(4-fluorophenyl)amino]piperidine-1-carbonyl}-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
(1R,5R)-6-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[2-(1H-indol-3-yl)ethyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
N-methyl-3-(pyridin-3-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
4-(1H-indazol-3-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(1H-imidazol-2-ylmethyl)-2-[(prop-2-en-1-yl)amino]benzamide
1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]cyclopropan-1-amine
N-[3-(4-{[2-(1H-indol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]-2-methoxybenzamide
{[2-(isoquinolin-1-yloxy)phenyl]methyl}dimethylamine
8-[2-(2-hydroxyethoxy)ethyl]-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one