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2-chloro-N-ethyl-4-[({1-oxaspiro[4.4]nonan-3-yl}carbamoyl)amino]benzamide
2-(2,8-dimethylquinoline-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-[(dimethylamino)methyl]-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-amino-7-hydroxy-4-(pyridin-4-yl)-5H,6H-benzo[h]quinoline-3-carbonitrile
7-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
8-[(3,4-difluorophenyl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-({4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
N-(but-2-yn-1-yl)-N-(furan-2-ylmethyl)-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
5-methyl-3-[5-(thiophene-3-sulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-1,2-oxazole
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-3-(2-methoxyphenyl)propan-1-one
6-[(2S)-1-acetylpyrrolidine-2-carbonyl]-1-methyl-3-(3-phenylphenyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-{[(1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)oxy]methyl}pyridine
2-cyclopentyl-9-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-4-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]pyridine
N-(2-phenylethyl)-3-{[1-(pyridin-3-ylmethyl)piperidin-4-yl]oxy}benzamide
1-[(3-fluorophenyl)methyl]-6-methyl-3-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-{[1-(2,5-difluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazol-5-amine
1-[2-methoxy-4-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
methyl 3-(3-methoxybenzamido)-5-{[2-(pyridin-2-ylsulfanyl)acetamido]methyl}benzoate
N-(2-hydroxyethyl)-1-(2-methoxyphenyl)-N-[(4-methylphenyl)methyl]-1H-pyrazole-4-carboxamide
N-({3-methyl-7-[2-(2-methyl-1H-indol-3-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
1-cyclopropanecarbonyl-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]piperidine-4-carboxamide
2-(2-fluorophenyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
2-[(2-hydroxyethyl)[3-(4H-1,2,4-triazol-4-yl)propyl]amino]ethan-1-ol
4-[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]pyridine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[1-(propan-2-yl)piperidine-4-carbonyl]piperazine
1-(2,6-dimethylhept-5-en-1-yl)-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
(1S,5R)-3-(4-aminopyridine-2-carbonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(oxolan-2-ylmethyl)propylamine
2-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}-1,3-benzoxazole
2-{4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-{[(4-fluorophenyl)methyl]sulfanyl}propanamide
(4aR,7aS)-1-methyl-4-(3-methyl-4-oxo-3,4-dihydrophthalazine-1-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(4-methoxyphenyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-2-(thiomorpholin-4-yl)pyridine-3-carboxamide
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]quinoline-8-sulfonamide
2-{4-[(5-chlorofuran-2-yl)methyl]morpholin-3-yl}acetic acid
N-cyclopropyl-1-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
1-ethyl-3-(2-methylpropyl)-N-(2,2,2-trifluoroethyl)-1H-pyrazole-5-carboxamide
(3aS,6aS)-2-[2-(6-methylpyridin-2-yl)ethyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-N-phenylpyrimidin-2-amine
N-(1,4-dioxan-2-ylmethyl)-N,1-dimethyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
4-hydroxy-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
5-fluoro-3-methyl-2-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}-1H-indole
4-(1H-indole-6-carbonyl)-1-(2-methylphenyl)piperazin-2-one
2-amino-4-(1H-indol-3-yl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-({[(3R,4R)-1-(2,5-difluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
4-{[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]oxy}pyridine
1-(2-chloro-3,5-difluorophenyl)-3-[(3-methyloxetan-3-yl)methyl]urea