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N-[(3R,4R)-3-hydroxy-1-(1H-indazole-3-carbonyl)piperidin-4-yl]pyridine-3-carboxamide
3-[4-(3-methylpiperidine-1-carbonyl)phenyl]-1-{2-[(pyridin-3-yl)amino]ethyl}urea
5-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-(methylsulfanyl)pyrimidine
2-cyclopentyl-8-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]propanamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-methyl-6-(propan-2-yl)-N-[(3,4,5-trimethoxyphenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-4-methyl-1,2,3-thiadiazole-5-carboxamide
2-(2-aminopyrimidin-5-yl)-N-ethyl-6-fluoro-N-(pyridin-2-ylmethyl)quinoline-4-carboxamide
N1-[1-(4-phenylphenyl)piperidin-4-yl]propane-1,3-diamine
N,6-dimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}quinolin-4-amine
3-(1-benzyl-1H-pyrazol-5-yl)-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-methylurea
8-(1-benzothiophen-2-ylmethyl)-1-ethyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(4-methanesulfonylphenyl)-6-(2-methyl-1H-imidazol-1-yl)pyridazine
1-{6-methylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-3-[3-(trifluoromethyl)benzoyl]piperidine
3-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-(4-methoxy-3,5-dimethylphenyl)urea
1-(2-fluorophenyl)-4-(4-{[3-(2-hydroxyethoxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)piperidin-4-ol
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
5-{2-oxo-2-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-2-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[(4-chlorophenyl)methyl]-8-[2-(ethylsulfanyl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
5-cyclobutyl-1-cyclohexyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
1-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-1,2,3,4-tetrahydroquinolin-2-one
1-methyl-3-[3-(pyridin-2-yl)azetidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
2-[2-methyl-3-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-indol-1-yl]acetamide
5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]pyridin-2-amine
3-[5-(ethylcarbamoyl)pyridin-2-yl]benzoic acid
1-{[1-(2-amino-5-ethyl-6-methylpyrimidin-4-yl)piperidin-3-yl]methyl}pyrrolidin-2-one
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-3-[(4-methylphenyl)formamido]propanamide
2-(azocan-1-yl)-1-{2,7-diazaspiro[4.5]decan-7-yl}ethan-1-one
2-[3-(1H-imidazol-1-yl)propyl]-9-(1-methylpiperidine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-ethyl-5-(3,6,7-trimethyl-1-benzofuran-2-yl)-1,2,4-oxadiazole
1-[(2-fluorophenyl)methyl]-4-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperazin-2-one
3-methyl-8-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
4-({3-[2-hydroxy-3-(piperidin-1-yl)propoxy]-4-methoxyphenyl}methyl)-1,4-diazepane-1-carbaldehyde
4-hydroxy-2-methyl-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
1-(2-{[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]amino}ethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
(1S,5R)-3-(2,4-dimethylpyrimidine-5-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1R,5R)-3-[1-(4-chlorophenyl)cyclobutanecarbonyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
8-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N3-[1-(3,5-difluorophenyl)cyclopropyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
({5-[1-(2-methoxypyridine-4-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
(2S,4R)-1-(naphthalen-1-ylmethyl)-N-(propan-2-yl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-(3,4-dichlorophenyl)-1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]ethan-1-one
2-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-ylmethyl]-4-hydroxyquinoline-6-carboxamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}pyridine-3-carboxamide
3-(2-amino-4-fluoro-1,3-benzothiazol-6-yl)-N,N-dimethylbenzamide
2-(2,5-dioxoimidazolidin-4-yl)-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}acetamide
6-(propan-2-yl)-2-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1H-indole