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3-[4-(5-methyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]-1,2-benzothiazole
2-[cyclohexyl(methyl)amino]-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]pyridine-3-carboxamide
2-(pyridin-3-yl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
5-chloro-N-[2-(2-fluorophenoxy)ethyl]pyridine-2-carboxamide
2-({imidazo[1,2-a]pyrimidin-2-ylformamido}methyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-(4-cyano-2-ethylphenyl)-3-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-3-methylurea
2-[3-(oxolan-3-yl)-5-(3-phenyl-1H-pyrazol-5-yl)-1H-1,2,4-triazol-1-yl]acetic acid
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-({[4-(dimethylamino)phenyl]methyl}amino)-N-methylpyrrolidine-2-carboxamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-6-methyl-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-(1-benzylpiperidin-4-yl)-3-(pyrrolidine-1-carbonyl)piperidine
N'-(adamantan-1-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}propanediamide
methyl 4-[2-(quinolin-2-yl)-1H-imidazol-1-yl]butanoate
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
(4S)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3,3,4-trimethylpiperidin-4-ol
{4-benzyl-1-[6-(propan-2-yl)pyridazin-3-yl]piperidin-4-yl}methanol
N-[1-(4-fluorophenyl)ethyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
N-(2-hydroxybutyl)-5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-[2-(4-fluorobenzenesulfonyl)ethyl]-3-[1-(propan-2-yl)-1H-pyrazol-4-yl]urea
3-({[(4-fluoro-3-methylphenyl)methyl]amino}methyl)-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-(pyrrolidin-3-yl)piperazine
5-(2-fluoro-6-methoxyphenyl)-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
3-(4-chlorobenzoyl)-1-(1H-imidazol-2-ylmethyl)piperidine
4-amino-2-[3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyrimidine-5-carbonitrile
N-(3-fluorophenyl)-1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-amine
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
6-methyl-2-[3-(trifluoromethoxy)phenyl]pyridine-3-carboxamide
2,6-dimethyl-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}imidazo[1,2-a]pyridine-3-carboxamide
7-(cyclopropylmethyl)-2-(4,4,4-trifluorobutanoyl)-2,7-diazaspiro[4.5]decan-6-one
N-[4-(4-methylbenzamido)phenyl]pyrazolo[1,5-a]pyridine-3-carboxamide
{6-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]pyridin-2-yl}methanol
7-[2-(4-phenylpiperidin-1-yl)acetyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1,4,6-trimethyl-3-[4-(oxolane-2-carbonyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
N-{1-[1-(2,3-difluorobenzoyl)piperidin-4-yl]-2-phenylethyl}-N,2-dimethylfuran-3-carboxamide
3-chloro-N-[(1-ethylpyrrolidin-2-yl)methyl]-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
(3S,4S)-4-cyclopropyl-1-[3-(3-fluorophenyl)propanoyl]pyrrolidine-3-carboxylic acid
ethyl 4-[(4-chlorophenyl)methyl]-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
1-[2-(dimethylamino)-2-(3-fluorophenyl)acetyl]piperidine-4-carbonitrile
6-[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidin-1-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
{2-[4-(3,5-dimethylfuran-2-carbonyl)morpholin-2-yl]ethyl}dimethylamine
4-{2-[1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)piperidin-2-yl]ethyl}phenol
(3S,4R)-N,N-dimethyl-1-[4-(morpholine-4-carbonyl)pyridin-2-yl]-4-(propan-2-yl)pyrrolidin-3-amine
N-[4-(pyridin-2-yl)butyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-(furan-2-yl)-5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}pyrimidine
1-{[1-(2-butyl-1,3-benzoxazole-5-carbonyl)piperidin-4-yl]methyl}pyrrolidin-2-one
2-cyclohexanecarbonyl-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-methyl-1-{[3-(methylsulfanyl)phenyl]methyl}pyrrolidine-3-carboxamide
9-(4-fluoro-2-methylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-ethyl-N,N-dimethyl-6-{4-[methyl(1,2-oxazol-3-ylmethyl)amino]piperidin-1-yl}pyrimidin-2-amine
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}isoquinoline