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N-methyl-3-(1,2-oxazinan-2-yl)-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]propanamide
N-cyclopropyl-2-(dimethylamino)-2-(4-fluorophenyl)-N-[(3-hydroxyphenyl)methyl]acetamide
1-(morpholin-4-yl)-2-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-{1-[2-(morpholin-4-yl)acetyl]piperidin-3-yl}benzoic acid
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-acetamidoacetamide
N-ethyl-5-[4-(morpholine-4-carbonyl)piperidine-1-carbonyl]pyrimidin-2-amine
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
2-(1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
N-(4-fluorophenyl)-1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-amine
4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
4-(3-{5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidine-1-carbonyl)-1,2-dihydrophthalazin-1-one
4-[(dimethylamino)methyl]-1-({4-[methyl(phenyl)amino]phenyl}methyl)piperidin-4-ol
3-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidine-1-carbonyl}-2-methylphenol
(4aS,8aS)-2-{1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-yl}-decahydroisoquinolin-4a-ol
methyl 1-(2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperidine-4-carboxylate
(2R)-N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]oxolane-2-carboxamide
2-[(4-chlorophenyl)methyl]-8-(3-methylpyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
N-[(3R,4S)-4-cyclopropyl-1-[3-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]-2-methoxyacetamide
N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-methyl-3-{[methyl(2,2,6,6-tetramethylpiperidin-4-yl)amino]methyl}-1H-indole-2-carboxylic acid
4-[1-(butan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-methyl-1H-pyrazole
2-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-2,7-diazaspiro[4.5]decan-6-one
1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
[1-(1-benzylpiperidin-4-yl)-3-[(2-methylphenyl)methyl]piperidin-3-yl]methanol
N-(1-cyclopropylethyl)-2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carboxamide
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
(3S,4R)-1-[2-(4-fluorophenyl)ethyl]-4-methylpiperidine-3,4-diol
methyl 3-{[3-(dimethylcarbamoyl)-2-methyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-7-carbonyl]amino}benzoate
N-benzyl-5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-(1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)piperidin-4-ol
5-(3-chlorophenyl)-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}-1,2,4-triazin-3-amine
ethyl 1-(5-acetylthiophene-2-carbonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
6-(4-methanesulfonylphenyl)-N,N-dimethylpyridazin-3-amine
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-N-(furan-2-ylmethyl)piperidine-4-carboxamide
5-chloro-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}pyridine-2-carboxamide
3-[2-(4-fluorophenyl)acetyl]-9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-3-(piperidin-3-yl)benzamide
methyl 4-{4-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]piperazin-1-yl}benzoate
7-({[(2-fluorophenyl)methyl]amino}methyl)-5-[2-(piperidin-1-yl)ethyl]-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N,1-dimethyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
4-(8-methoxy-2H-chromen-3-yl)-1-methyl-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-(5-amino-4-phenyl-1H-pyrazole-3-carbonyl)morpholine-2-carboxylic acid
2-(6-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]acetamide
3-[({[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]carbamoyl}amino)methyl]-1,2,4-oxadiazole-5-carboxamide
N-(2-methylprop-2-en-1-yl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
8-(1H-indol-3-ylmethyl)-1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-ethylpyrimidine-5-carboxamide
1-[2-(1H-imidazol-5-yl)ethyl]-5-(4-methyl-1,3-oxazol-5-yl)-3-(phenoxymethyl)-1H-1,2,4-triazole