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4-(cyclohexylmethyl)-3-[2-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}pyrimidin-2-amine
N-[(3S,5S)-1-(2,5-dimethylfuran-3-carbonyl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
1-(adamantan-2-yl)-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
(2R)-2-amino-2-cyclohexyl-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
3-(3-methylbut-2-en-1-yl)-1-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]piperidine-3-carboxylic acid
N-cyclopentyl-2-[(3,4-dimethoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
2-(hydroxymethyl)-N-[2-(2-phenoxyethoxy)phenyl]azepane-1-carboxamide
N-{1-[2-(2-methoxyethyl)-1,3-benzoxazole-6-carbonyl]pyrrolidin-3-yl}acetamide
1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(2-phenylethyl)piperidine
1-cyclopentyl-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-methyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
3-{[(2-methoxyethyl)[(4-methylphenyl)methyl]amino]methyl}-4H-chromen-4-one
1-{2,7-diazaspiro[4.5]decan-7-yl}-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-[2-(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]acetamide
5-fluoro-2-(1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
4-{5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(cyclohex-1-en-1-ylmethyl)-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
1-(2-amino-6-methylpyrimidin-4-yl)-4-cyclobutanecarbonyl-1,4-diazepan-6-ol
5-(2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one
N-(2-methoxyethyl)-3,5-dimethyl-4-oxo-N-(1,3-thiazol-2-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-5-methyl-1,3,4-oxadiazol-2-amine
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
2-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-[4-(piperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[3-(1,2-oxazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3-(piperidin-1-yl)pyridine
(3R,4R)-1-[1-(4-fluorophenyl)piperidin-4-yl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole
[(2-methoxypyrimidin-5-yl)methyl](methyl){2-[(4-methylphenyl)sulfanyl]ethyl}amine
3-{2-azabicyclo[2.2.1]heptan-2-ylmethyl}-1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-1,2-dihydroquinolin-2-one
3-{[3-(1H-imidazol-1-yl)propyl]amino}-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
4-[4-(2-ethylpyrimidine-5-carbonyl)piperazine-1-carbonyl]morpholine
2-(1-ethylpiperidin-4-yl)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]acetamide
(2S,4S)-N,N-diethyl-4-[1-(2-fluorophenyl)cyclopropaneamido]-1-methylpyrrolidine-2-carboxamide
N-ethyl-2-(2-methoxyquinolin-3-yl)benzamide
N4-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
7-(2-phenoxybutanoyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(5-methoxyfuran-2-carbonyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(propan-2-yl)-9-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
7-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
1-[(4-methyl-1H-imidazol-5-yl)methyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
methyl(oxolan-3-ylmethyl)[(2-phenyl-1,3-thiazol-4-yl)methyl]amine
3-{[(1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)oxy]methyl}pyridine
4-[2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,4-oxazepane
3-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[({[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}amino)methyl]piperidin-3-ol
5-[3-(dimethylamino)phenyl]-1H-indazol-3-amine
1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
1-[(5-methylthiophen-2-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide