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3-(3-chlorophenyl)-1-(4-methylpiperazin-1-yl)-3-phenylpropan-1-one
(1-{1-tert-butyl-3-[(3,4-dimethoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}propan-2-yl)dimethylamine
1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-{4-[3-({[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
1-(2-phenylethyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
2-(2-{[3-(hydroxymethyl)-3-methylpiperidin-1-yl]methyl}-4-(pyrimidin-2-yl)phenoxy)acetic acid
{1-[({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)methyl]cyclobutyl}methanol
4-[2-(thiophen-2-yl)pyrimidine-5-carbonyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-6-azaspiro[2.5]octane
2-(2-methyl-1H-indol-3-yl)-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetamide
2-{4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
N-(4-ethoxy-2-fluorophenyl)-4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carboxamide
5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-(3-{[(3-hydroxypropyl)(methyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3-[2-(4-fluorophenyl)morpholine-4-carbonyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
N-[(1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperidin-4-yl)methyl]acetamide
4-[(2-chlorophenyl)methyl]-1-(4-phenylbenzoyl)-1,4-diazepan-5-one
4-(1-{[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]amino}ethyl)hepta-1,6-dien-4-ol
N,2-dimethyl-N-[(1-methylpiperidin-2-yl)methyl]-3-[(pyridin-2-ylmethyl)amino]benzamide
3-(3-{3,9-diazaspiro[5.5]undecan-3-ylmethyl}-1H-indol-1-yl)propanoic acid
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(1H-pyrrole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1R,3S)-7-[2-hydroxy-6-(trifluoromethyl)pyridine-3-carbonyl]-7-azaspiro[3.5]nonane-1,3-diol
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
4-[(dimethyl-1,2-oxazol-4-yl)methyl]-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[3-(1H-indol-1-yl)propyl]-1-(oxolane-2-carbonyl)piperidin-4-amine
N-[1-(4-methanesulfonylphenyl)ethyl]-2-methyl-4-phenylpyridine-3-carboxamide
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-cyclobutanecarbonylpiperidine
1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,2,3,4-tetrahydroquinolin-2-one
6-[1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]-3,4-dihydropyrimidin-4-one
1-(4-phenyl-1H-imidazole-5-carbonyl)azepan-4-amine
1,6-dimethyl-3-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-(cyclopropylmethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[2-(pyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
2-methoxy-1-{4-[3-(methylsulfanyl)butyl]-1,4-diazepan-1-yl}ethan-1-one
1-[(2,3-dimethoxyphenyl)methyl]-4-[(2-methoxyphenyl)methyl]piperazine
(7S,8aS)-7-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)amino]-2-methyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-methoxy-5-[4-(thiophen-2-yl)-1H-imidazol-1-yl]pyridine
N-ethyl-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-3-carboxamide
(4aS,8aR)-6-[3-(3-fluorophenyl)propanoyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
6-(2-chlorophenyl)-2-(4-fluoropiperidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-(2-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,3,6-trimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
3-[(dimethylamino)methyl]-1-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]piperidin-3-ol
6-(2-acetylphenyl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
1-({5-[(2S)-4,4-difluoropyrrolidine-2-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,5-dihydro-1H-pyrrole
5-fluoro-N4,N4-dimethyl-N2-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]pyrimidine-2,4-diamine
1-{3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-2-(methoxymethyl)piperidine
(4aR,8aR)-2-(1-benzofuran-5-carbonyl)-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
[(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)methyl](methyl)amine