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N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-1H-1,2,3-triazole-5-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)amine
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-{methyl[(3-methylpyridin-4-yl)methyl]amino}acetic acid
[1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
4-(3-phenylbutyl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]-3-propanamidobenzamide
N-[(2-methoxyphenyl)methyl]-4,5-dimethyl-N-propylthiophene-2-carboxamide
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
N-[1-(6-cyclopropylpyrimidin-4-yl)pyrrolidin-3-yl]acetamide
N-[(1R)-1-(4-methoxyphenyl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
[(3R,4R)-1-[(4-fluoro-3-methylphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-{5H,6H-benzo[h]quinazolin-2-yl}-N-(2-hydroxyethyl)-5-methyl-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-{[1-(2-phenylethyl)piperidin-3-yl]methyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-benzyl-N-(3-hydroxy-2-methylpropyl)-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-[(1S)-1-cyclohexylethyl]-4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
1-(1,2,5-thiadiazole-3-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
N-[1-(1H-indol-2-yl)ethyl]-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
2-[(1-ethyl-1H-indol-4-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-[3-(pyridin-4-yl)propyl]cyclopentane-1,3-dicarboxamide
4-hydroxy-N-methyl-N-[3-(2-methylphenoxy)propyl]-2-phenylpyrimidine-5-carboxamide
ethyl 5-({[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}methyl)-1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-1H-pyrazole-4-carboxylate
N,N-dimethyl-2-(pyridin-4-yl)-7-[(2R)-pyrrolidine-2-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
[(3R,4R)-1-(3-chloro-5-fluorobenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-cyclohexyl-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
1-{4-[4-(2,6-dimethoxypyrimidin-4-yl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
3-(furan-3-ylmethyl)-1-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
1-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-(pyridin-2-ylmethyl)-1,4-diazepane
(2R,3R,6R)-5-(5-chloropyridine-3-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(1-{1-[(3,5-dichloropyridin-4-yl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
N-(5-methoxy-2-methylphenyl)-4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carboxamide
1-(2-methoxyethyl)-4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
6-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
3-{1-[(2,2-dimethyloxan-4-yl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(4-fluorophenyl)methyl]piperidine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-6-(4-methylpiperazine-1-carbonyl)pyrazin-2-amine
ethyl 1-({2-[benzyl(methyl)carbamoyl]imidazo[1,2-a]pyridin-3-yl}methyl)piperidine-3-carboxylate
3-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-1-(4-methoxy-3,5-dimethylphenyl)urea
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidin-4-yl}propanamide
7-(5-chloropyridin-2-yl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(azetidine-1-carbonyl)-5-chloro-3-methyl-1H-indole
6-methyl-1-{3-[4-(3-methylphenoxy)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
3-(diphenylmethyl)-5-methanesulfonyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-benzyl-9-(4-oxo-4-phenylbutyl)-2,9-diazaspiro[5.5]undecan-3-one
8-acetyl-2-(1H-indol-5-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
9-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-6-(4-methoxyphenyl)-6,9-diazaspiro[4.5]decan-7-one
(2-methoxyethyl)(methyl){[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}amine