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3-[2-fluoro-3-(pyrrolidin-1-ylmethyl)phenoxy]-2,5-dimethylpyrazine
[(3-ethoxy-4-methoxyphenyl)methyl](methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
(3S,4R)-4-(2-methoxyphenyl)-1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}pyrrolidine-3-carboxylic acid
2-[2-({3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
4-phenyl-1-[6-(pyridin-3-yl)pyridine-3-carbonyl]azepane
N-({7-[(2E)-3-(4-chlorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(1H-imidazol-1-yl)acetamide
5-{[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-N-propylpyrimidin-2-amine
2-(3-fluorophenyl)-1-(4-methyl-1H-imidazole-2-carbonyl)piperidine
3-chloro-2-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)-1H-indole
1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-4-(pyrrolidin-1-yl)piperidine
1-benzyl-4-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperazin-2-one
3-(1,3-benzothiazol-6-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
methyl[(5-phenyl-1,2-oxazol-3-yl)methyl]{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
3-({2-[1-(2-fluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
4-fluoro-N-[2-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]benzamide
1-({[2-(hydroxymethyl)quinazolin-4-yl]amino}methyl)cyclohexan-1-ol
3-(2-methoxyethyl)-1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]piperidine-3-carboxylic acid
2-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-methyl-7-oxo-N-[2-(pyridin-2-yl)ethyl]-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
5-({3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
3-(4-chloro-1H-pyrazol-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}propanamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamide
2-{2-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}propanamide
(2S)-1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-phenylbutan-1-one
2-(1-benzyl-4-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperazin-2-yl)ethan-1-ol
N-cyclopentyl-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(1,3-benzoxazol-2-ylmethyl)-N-methyl-1-benzofuran-5-carboxamide
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]propan-1-one
N-ethyl-1-{2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}pyrrolidine-3-carboxamide
N-cyclopropyl-3-[5-(2-phenoxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
N-[3-(dimethylamino)-2,2-dimethylpropyl]-4-[ethyl(2-methylprop-2-en-1-yl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)({[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
6-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(3-methoxyphenyl)-1-(pyridin-2-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)propyl]pyridine-4-carboxamide
1-(5-{[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
(3S,4R)-4-(2-methoxyphenyl)-1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrrolidine-3-carboxylic acid
2-[4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carbonyl]benzonitrile
1-{5-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]thiophen-2-yl}ethan-1-one
N-(1H-imidazol-2-ylmethyl)-N,2-dimethyl-6-(piperidin-4-yl)pyrimidin-4-amine
1-(3-ethylphenyl)-3-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}urea
N-(6-ethylpyridin-2-yl)-3-[(2-methyl-5-oxo-1,4-diazepan-1-yl)methyl]benzamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-4-yl]propanamide
[4-(4-{1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl}pyridin-2-yl)phenyl]methanol
1-{5-[(2-aminopyrimidin-4-yl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-ol
N-{5-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]quinolin-8-yl}acetamide
methyl 2-[3-(3-oxopiperazine-1-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetate
1-[4-(azetidin-1-ylmethyl)-2-methoxyphenoxy]-3-(azocan-1-yl)propan-2-ol