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1-[3-(5-methylfuran-2-yl)benzoyl]pyrrolidin-3-ol
(5S)-5-{[({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(pyridin-4-ylmethyl)amino]methyl}pyrrolidin-2-one
N-cyclopropyl-3-(3-methyl-1H-pyrazol-1-yl)-N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}propanamide
2,6-diamino-4-(4-chloro-1-methyl-1H-indazol-3-yl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
(3aR,6aR)-2-ethyl-5-(5-methoxypyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[3-oxo-3-(pyrrolidin-1-yl)propyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
2-(5-ethyl-1-benzofuran-3-yl)-1-[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
9-(1H-imidazol-2-ylmethyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N4-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidine-4,6-diamine
1-butyl-3-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-1-(pyridin-4-ylmethyl)urea
6-[3-(3-methoxyphenoxy)azetidin-1-yl]pyridine-2-carboxylic acid
4-({5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,2,4-oxadiazol-3-yl}methyl)-1-propylpiperidine
1-cyclobutanecarbonyl-4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}piperidine
1-(4-methoxyphenyl)-3-methyl-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperazin-2-one
3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(4-sulfamoylphenyl)urea
1-(diethylamino)-3-[2-methoxy-4-({[2-(piperidin-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(quinoxaline-6-carbonyl)pyrrolidin-3-yl]methanol
5-({4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-3-carbonyl]-1,3-oxazol-2-yl}methoxy)isoquinoline
1-(cyclohexylmethyl)-N3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-{5-oxo-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-4-yl}propanoic acid
3-[2-(diethylamino)ethyl]-3-ethyl-1-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}urea
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
3-[(3S,4R)-1-benzyl-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-[2-(diethylamino)ethyl]propanamide
2-(4-cyanophenyl)-2-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}acetic acid
2-(2,3-dihydro-1H-inden-1-yl)-N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
2-(1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}azetidin-3-yl)pyridine
2-(2H-1,3-benzodioxol-5-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
N-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
4-(4-chlorophenoxy)-4-(2,5-dihydro-1H-pyrrole-1-carbonyl)piperidine
N-ethyl-1-[(2-fluorophenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
(1R,3S,5S)-8-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane
1-[(2S)-2-amino-3-(1H-imidazol-4-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(3-chlorophenoxy)-N-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]propanamide
2-{2-[4-(cyclopropylmethyl)piperazin-1-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(3R,4S)-4-cyclopropyl-1-(2,4-dimethylpyrimidine-5-carbonyl)pyrrolidin-3-amine
(3R,4R)-3-cyclobutyl-4-methyl-1-(1,3-thiazol-2-ylmethyl)pyrrolidin-3-ol
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-[3-(1H-imidazol-1-yl)propyl]pyridin-2-amine
1-(4-{[1-(1H-imidazol-2-yl)ethyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
7-methanesulfonyl-N-[2-(1,3-thiazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(2R)-2-cyclohexyl-N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-hydroxyacetamide
1-{2,7-diazaspiro[4.5]decan-2-yl}-2-(2-methoxyethoxy)ethan-1-one
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopent-1-ene-1-carboxamide
3-({4-[1-(3,5-dimethylfuran-2-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
6-methyl-4-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
6-tert-butyl-3-(3-hydroxybutyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
2-(3-fluorophenyl)-1-(oxane-4-carbonyl)piperidine
1-(2-chlorophenyl)-4-(3-fluoro-4-methylbenzoyl)-5-methylpiperazin-2-one
N-[(3S,5S)-1-(cyclopentylmethyl)-5-(diethylcarbamoyl)pyrrolidin-3-yl]-2-methyl-1H-pyrrole-3-carboxamide